SCHEMBL2362023

SCHEMBL2362023

COC(=O)c1ccc2[nH]c(-c3c(F)cccc3Cl)nc2c1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RHEB Q15382 1/20 0.57
PTGES O14684 6/20 0.49
KDM4E B2RXH2 3/20 0.48
ALDH1A1 P00352 3/20 0.48
LMNA P02545 2/20 0.48
NPC1 O15118 1/20 0.48
PKM P14618 1/20 0.48
HPGD P15428 1/20 0.48
NFKB1 P19838 1/20 0.48
RAB9A P51151 1/20 0.48
NFKB2 Q00653 1/20 0.48
RELA Q04206 1/20 0.48
SMN1; SMN2 Q16637 1/20 0.48
DGAT1 O75907 2/20 0.46
JAK2 O60674 2/20 0.43
TYK2 P29597 1/20 0.43
MAPK14 Q16539 1/20 0.43
MMP2 P08253 1/20 0.42
MMP9 P14780 1/20 0.42
MMP8 P22894 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361214 0.91 CSNK1E (0.52) RHEBKDM4EALDH1A1NPC1PKM
SCHEMBL2361289 0.89 DGAT1 (0.48) RHEBPTGESDGAT1TP53
SCHEMBL2360771 0.86 PTGES (0.50) PTGESKDM4EALDH1A1NPC1HPGD
SCHEMBL2361432 0.85 KDM4E (0.47) RHEBPTGESKDM4EALDH1A1LMNA
SCHEMBL2362063 0.84 KDM4E (0.47) RHEBPTGESKDM4EALDH1A1LMNA
SCHEMBL2361142 0.84 DGAT1 (0.44) RHEBPTGESLMNANPC1RAB9A
SCHEMBL2361818 0.83 RAB9A (0.47) RHEBPTGESKDM4EALDH1A1LMNA
SCHEMBL1251886 0.82 DGAT1 (0.65) RHEBKDM4EALDH1A1LMNANPC1
SCHEMBL2361754 0.82 PRSS12 (0.56) PTGESKDM4EALDH1A1NPC1RAB9A
SCHEMBL2361026 0.81 DGAT1 (0.41) RHEBPTGESALDH1A1NPC1RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed