SCHEMBL2361495

SCHEMBL2361495

CCCCc1nc(N)c2c(-c3ccc(C)cc3)n[nH]c2n1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 5/20 0.40
ALDH1A1 P00352 3/20 0.40
GAA P10253 1/20 0.40
NPC1 O15118 1/20 0.39
TP53 P04637 1/20 0.39
TSHR P16473 1/20 0.39
RAB9A P51151 1/20 0.39
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ADORA1 P30542 2/20 0.36
ADORA3 P0DMS8 1/20 0.36
TLR8 Q9NR97 1/20 0.35
MAPK1 P28482 2/20 0.34
PIK3CD O00329 1/20 0.34
PIK3CA P42336 1/20 0.34
PIK3CB P42338 1/20 0.34
PIK3CG P48736 1/20 0.34
PRKDC P78527 1/20 0.34
HPGD P15428 2/20 0.33
ADORA2A P29274 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5066107 0.85 TLR8 (0.40) SMN1; SMN2NPC1TP53TSHRRAB9A
SCHEMBL5067787 0.80 EPHA4 (0.41) SMN1; SMN2NPC1TP53TSHRRAB9A
SCHEMBL5748863 0.76 MEN1 (0.42) SMN1; SMN2ALDH1A1TP53RAB9AMEN1
SCHEMBL3782102 0.72 PIK3CD (0.57) SMN1; SMN2ALDH1A1TP53TSHRMEN1
SCHEMBL17505368 0.71 BTK (0.46) PIK3CDPIK3CAPIK3CBPIK3CGPRKDC
SCHEMBL28827843 0.68 ADORA3 (0.45) SMN1; SMN2ALDH1A1GAANPC1TSHR
SCHEMBL12713498 0.66 PIK3CD (0.50) ALDH1A1TP53TSHRMEN1KMT2A
SCHEMBL7540624 0.65 XDH (0.42) ALDH1A1ADORA1ADORA3ADORA2AADORA2B
SCHEMBL15020484 0.64 DPP4 (0.43) SMN1; SMN2ALDH1A1GAANPC1TP53
SCHEMBL2318766 0.64 GPR84 (0.47) ALDH1A1GAAADORA3HPGDADORA2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358720-A2 FUSED RING HETEROARYL KINASE INHIBITORS The Regents of the University of California (US) 2011-08-24 EP disclosed
WO-2010045542-A2 FUSED RING HETEROARYL KINASE INHIBITORS THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2010-04-22 WO disclosed