SCHEMBL2361706

SCHEMBL2361706

COc1cc(N)cc2nc(-c3c(F)cccc3Cl)[nH]c12

nearest known ligand 0.48

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
PTGES O14684 16/20 0.48
JAK2 O60674 1/20 0.47
PDE7A Q13946 2/20 0.47
CYP2D6 P10635 1/20 0.40
CYP2C9 P11712 1/20 0.40
ORAI1 Q96D31 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2361612 0.82 PTGES (0.50) PTGESJAK2CYP2D6CYP2C9
SCHEMBL2361351 0.81 AMY1A (0.45) PTGESJAK2CYP2D6CYP2C9
SCHEMBL2361320 0.75 PTGES (0.47) PTGESJAK2CYP2C9
SCHEMBL5202015 0.74 RPS6KA2 (0.45) PTGESJAK2
SCHEMBL2361007 0.74 PTGES (0.61) PTGESJAK2CYP2D6CYP2C9
SCHEMBL2362277 0.73 PLAU (0.51)
SCHEMBL2361085 0.72 AMY1A (0.44) PTGESJAK2PDE7AORAI1
SCHEMBL2361888 0.72 AMY1A (0.47) PTGESJAK2PDE7ACYP2D6CYP2C9
SCHEMBL14629876 0.72 PTGES (0.52) PTGESJAK2CYP2C9
SCHEMBL2361818 0.72 RAB9A (0.47) PTGES

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011099832-A2 NOVEL BENZIMIDAZOLE COMPOUND, PREPARATION METHOD THEREOF AND PHARMACEUTICAL COMPOSITION COMPRISING THE SAME CRYSTALGENOMICS, INC. (KR) 2011-08-18 WO disclosed