SCHEMBL23618989

SCHEMBL23618989

CCSc1ccc(CNC(=O)c2ccc3c(c2)OCC(C(C)C)N3c2cccc(C(F)(F)F)c2)cc1

nearest known ligand 0.41

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 2/20 0.40
DDR1 Q08345 1/20 0.40
RORC P51449 2/20 0.39
PPARG P37231 1/20 0.39
HTR7 P34969 1/20 0.39
DRD2 P14416 1/20 0.38
MLYCD O95822 1/20 0.37
PSEN1 P49768 1/20 0.37
PSEN2 P49810 1/20 0.37
APH1B Q8WW43 1/20 0.37
NCSTN Q92542 1/20 0.37
APH1A Q96BI3 1/20 0.37
PSENEN Q9NZ42 1/20 0.37
CCR2 P41597 2/20 0.36
SERPINE1 P05121 1/20 0.36
ELANE P08246 1/20 0.36
KLKB1 P03952 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23619016 0.92 ROCK2 (0.44) ROCK2RORCPPARGDRD2
SCHEMBL28623367 0.80 HTR7 (0.43) HTR7CCR2SERPINE1
SCHEMBL28627879 0.79 LMNA (0.42)
SCHEMBL23619064 0.75 MAPT (0.43) DDR1RORC
SCHEMBL23619005 0.75 ROCK2 (0.45) ROCK2PPARGDRD2
SCHEMBL23619025 0.73 ROCK2 (0.45) ROCK2PPARGDRD2
SCHEMBL23619113 0.73 ROCK2 (0.45) ROCK2RORCPPARGDRD2
SCHEMBL23618986 0.72 RORC (0.37) RORC
SCHEMBL28626446 0.72 RORC (0.37) RORC
SCHEMBL23619094 0.72 ROCK2 (0.44) ROCK2PPARGDRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021136339-A1 AMIDE COMPOUND WITH BICYCLIC STRUCTURE AND USE THEREOF IN DRUG 广东东阳光药业有限公司 2021-07-08 WO disclosed