SCHEMBL28627879

SCHEMBL28627879

COC(=O)c1ccc2c(c1)OCC(C(C)C)N2c1cccc(C(F)(F)F)c1

nearest known ligand 0.42

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.42
PHGDH O43175 1/20 0.41
IDH1 O75874 2/20 0.40
ACACB O00763 2/20 0.39
HSD17B10 Q99714 1/20 0.39
KCNN4 O15554 1/20 0.39
NPSR1 Q6W5P4 2/20 0.38
CACNA1B Q00975 1/20 0.38
KMT2A Q03164 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 2/20 0.37
GUSB P08236 1/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
TP53 P04637 1/20 0.37
CACNA1F O60840 1/20 0.36
CACNA1D Q01668 1/20 0.36
CACNA1S Q13698 1/20 0.36
CACNA1C Q13936 1/20 0.36
PABPC1 P11940 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28623367 0.89 HTR7 (0.43) LMNAIDH1ACACBKMT2AMEN1
SCHEMBL28629894 0.89 IDH1 (0.38) LMNAIDH1
SCHEMBL23618989 0.79 ROCK2 (0.40)
SCHEMBL28618410 0.78 TEAD1 (0.39) IDH1KMT2AMEN1MAPT
SCHEMBL28626446 0.75 RORC (0.37) ACACBNPSR1
SCHEMBL23618986 0.75 RORC (0.37) ACACBNPSR1
SCHEMBL17991562 0.74 PHGDH (0.41) LMNAPHGDHCACNA1BKMT2AMEN1
SCHEMBL29501141 0.74 PHGDH (0.41) LMNAPHGDHCACNA1BKMT2AMEN1
SCHEMBL5854429 0.74 P2RX3 (0.50) IDH1TP53
SCHEMBL5854432 0.74 P2RX3 (0.50) IDH1TP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-113121463-A Amide compound with bicyclic structure and application thereof in medicines 广东东阳光药业有限公司 2021-07-16 CN disclosed