SCHEMBL2364035

SCHEMBL2364035

Nc1ncccc1C(=O)OC(=O)c1ccccc1OC(F)(F)F

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
NAPRT Q6XQN6 1/20 0.46
PRKCI P41743 2/20 0.43
KDM4E B2RXH2 1/20 0.43
ALDH1A1 P00352 1/20 0.43
DHODH Q02127 1/20 0.41
SCN10A Q9Y5Y9 3/20 0.40
ATR Q13535 1/20 0.40
HCRTR1 O43613 1/20 0.40
HCRTR2 O43614 1/20 0.40
CDK2 P24941 1/20 0.39
KCNK3 O14649 3/20 0.39
KCNK9 Q9NPC2 3/20 0.39
TLR7 Q9NYK1 2/20 0.39
FFAR4 Q5NUL3 1/20 0.38
SCN5A Q14524 1/20 0.37
SCN9A Q15858 1/20 0.37
SCN2A Q99250 1/20 0.37
SCN3A Q9NY46 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20561089 0.84 KCNK3 (0.49) ALDH1A1HCRTR1HCRTR2KCNK3KCNK9
SCHEMBL219458 0.82 NAPRT (0.66) NAPRTPRKCIKDM4EALDH1A1
SCHEMBL20561090 0.77 SLC6A3 (0.47) ALDH1A1SCN10AKCNK3KCNK9FFAR4
SCHEMBL2303054 0.76 LTA4H (0.49) NAPRTSCN10AATRTLR7SCN9A
Hydrochloric Acid SCHEMBL28016225 0.76 SLC6A3 (0.46) ALDH1A1SCN10AKCNK3KCNK9FFAR4
SCHEMBL28016834 0.74 HSD11B1 (0.52) ALDH1A1CDK2KCNK3KCNK9FFAR4
Hydrochloric Acid SCHEMBL29857909 0.74 LTA4H (0.47) NAPRTSCN10AATRTLR7SCN9A
SCHEMBL7542152 0.73 CDK2 (0.44) NAPRTDHODHSCN10AATRHCRTR1
SCHEMBL28016181 0.72 MGLL (0.54) KCNK3KCNK9FFAR4
SCHEMBL12951000 0.72 NAPRT (0.56) NAPRTPRKCIKDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2358202-A1 BENZIMIDAZOLE AND AZA-BENZIMIDAZOLE CARBOXAMIDES Merck Sharp & Dohme Corp. (US) 2011-08-24 EP disclosed