SCHEMBL23645387

SCHEMBL23645387

COc1ccc(COC2CCn3nc(C(=O)O)cc3OC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 4/20 0.39
RAB9A P51151 2/20 0.39
NPC1 O15118 1/20 0.39
POLB P06746 1/20 0.39
KDM5A P29375 1/20 0.38
KDM4C Q9H3R0 1/20 0.38
KDM5B Q9UGL1 1/20 0.38
ALDH1A1 P00352 3/20 0.38
CYP1A2 P05177 1/20 0.38
CYP2C19 P33261 1/20 0.38
HPGD P15428 2/20 0.37
KDM4E B2RXH2 3/20 0.37
MAPT P10636 1/20 0.37
NAAA Q02083 1/20 0.36
ASPH Q12797 1/20 0.36
RIOX2 Q8IUF8 1/20 0.36
KDM8 Q8N371 1/20 0.36
MGLL Q99685 3/20 0.36
FAAH O00519 1/20 0.36
RPA1 P27694 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23645404 0.89 TP53 (0.41) SMN1; SMN2RAB9ANPC1POLBALDH1A1
SCHEMBL23645395 0.77 MGLL (0.37) KDM4EMGLL
SCHEMBL23645383 0.67 KMT2A (0.39) POLBALDH1A1CYP2C19HPGDKDM4E
SCHEMBL21626249 0.67 CARM1 (0.43) ALDH1A1CYP2C19NAAALMNAHRH3
SCHEMBL23645400 0.65 RBP4 (0.34) ALDH1A1KDM4E
SCHEMBL17011149 0.64 RAB9A (0.52) SMN1; SMN2RAB9ANPC1POLBKDM5A
SCHEMBL21331023 0.64 PDK1 (0.39) SMN1; SMN2POLBALDH1A1KDM4EMGLL
SCHEMBL14800401 0.64 ALDH1A1 (0.44) SMN1; SMN2RAB9AALDH1A1HPGDKDM4E
SCHEMBL4494006 0.64 ALDH1A1 (0.82) SMN1; SMN2RAB9ANPC1POLBALDH1A1
SCHEMBL23645447 0.64 KMT2A (0.40) POLBALDH1A1HPGDKDM4EMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12421225-B2 Heteroaromatic amide derivative and medicament containing the same KAKEN PHARMACEUTICAL CO., LTD. (JP) 2025-09-23 US disclosed
CN-112689636-B Novel heteroatom aromatic amide derivative and pharmaceutical agent containing same 科研制药株式会社 2024-08-20 CN disclosed
EP-3851436-B1 NOVEL HETEROAROMATIC AMIDE DERIVATIVE AND MEDICINE CONTAINING SAME KAKEN PHARMA CO LTD (JP) 2024-06-12 EP disclosed
US-20230086366-A1 Novel heteroaromatic amide derivative and medicament containing the same KAKEN PHARMACEUTICAL CO., LTD. (JP) 2023-03-23 US disclosed
EP-3851436-A1 NOVEL HETEROAROMATIC AMIDE DERIVATIVE AND MEDICINE CONTAINING SAME Kaken Pharmaceutical Co., Ltd. (JP) 2021-07-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230086366-A1 Novel heteroaromatic amide derivative and medicament containing the same SCN7A, HCN4, SCN4A SMN1; SMN2 2354/4885RAB9A 1336/4885NPC1 1097/4885
US-12421225-B2 Heteroaromatic amide derivative and medicament containing the same SCN7A, HCN4, SCN4A SMN1; SMN2 2261/4885RAB9A 1727/4885NPC1 1165/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.