SCHEMBL23647557

SCHEMBL23647557

COc1ccc(C2(N)CCN(C(=O)O)CC2)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.51
TET3 O43151 2/20 0.51
FBXL19 Q6PCT2 2/20 0.51
CXXC5 Q7LFL8 2/20 0.51
TET1 Q8NFU7 2/20 0.51
KDM2B Q8NHM5 2/20 0.51
CXXC4 Q9H2H0 2/20 0.51
KDM2A Q9Y2K7 2/20 0.51
CYP3A4 P08684 3/20 0.46
CYP2C19 P33261 1/20 0.46
POLB P06746 1/20 0.45
SMN1; SMN2 Q16637 4/20 0.44
USP2 O75604 2/20 0.44
ALDH1A1 P00352 1/20 0.44
CYP2C9 P11712 2/20 0.43
MAPK1 P28482 1/20 0.43
HIF1A Q16665 1/20 0.43
CYP2D6 P10635 2/20 0.43
HPGD P15428 1/20 0.43
CYP1A2 P05177 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23381801 0.84 KMT2A (0.44) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL16874836 0.83 OPRM1 (0.59) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL23647376 0.82 KMT2A (0.59) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL13908097 0.82 BACE1 (0.55) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL10322683 0.80 OPRM1 (0.47) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL4662764 0.80 CA12 (0.43) SMN1; SMN2ALDH1A1HPGDOPRM1OPRD1
SCHEMBL1581919 0.79 OPRM1 (0.56) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL23647460 0.78 ALDH1A1 (0.54) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL16874714 0.78 HSD11B1 (0.56) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL895814 0.78 MAOB (0.52) CYP3A4ALDH1A1MAPK1MAPTOPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021143680-A1 HETEROARYL DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江海正药业股份有限公司 2021-07-22 WO disclosed