SCHEMBL23647376

SCHEMBL23647376

COc1ccc(C2(C(N)=O)CCN(C(=O)O)CC2)cc1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 3/20 0.59
TET3 O43151 2/20 0.59
FBXL19 Q6PCT2 2/20 0.59
CXXC5 Q7LFL8 2/20 0.59
TET1 Q8NFU7 2/20 0.59
KDM2B Q8NHM5 2/20 0.59
CXXC4 Q9H2H0 2/20 0.59
KDM2A Q9Y2K7 2/20 0.59
CYP3A4 P08684 1/20 0.50
CYP2C19 P33261 1/20 0.50
TACR2 P21452 4/20 0.49
TACR1 P25103 4/20 0.49
LMNA P02545 1/20 0.46
F10 P00742 1/20 0.44
CHRM5 P08912 2/20 0.44
CHRM3 P20309 2/20 0.44
CHRM1 P11229 1/20 0.44
OPRM1 P35372 1/20 0.43
OPRL1 P41146 1/20 0.43
HRH3 Q9Y5N1 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1480336 0.85 LMNA (0.55) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL23660780 0.83 BACE1 (0.53) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL23647557 0.82 KMT2A (0.51) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL10002472 0.82 LMNA (0.60) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL5205623 0.82 LMNA (0.65) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL16874836 0.81 OPRM1 (0.59) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL2112323 0.80 LMNA (0.68) KMT2ACYP3A4CYP2C19LMNACHRM1
SCHEMBL23647652 0.80 NNMT (0.43) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL23647525 0.78 HSD11B1 (0.40) KMT2ATET3FBXL19CXXC5TET1
SCHEMBL2701584 0.78 ALDH1A1 (0.59) KMT2ACYP3A4CYP2C19LMNAHRH3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021143680-A1 HETEROARYL DERIVATIVE, PREPARATION METHOD THEREFOR, AND USE THEREOF 浙江海正药业股份有限公司 2021-07-22 WO disclosed