SCHEMBL236515

SCHEMBL236515

COc1ccccc1CC(=O)c1ccc(O)cc1O

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 1.00
ALDH1A1 P00352 4/20 0.63
MAPK1 P28482 2/20 0.63
HPGD P15428 3/20 0.58
MEN1 O00255 3/20 0.58
KMT2A Q03164 3/20 0.58
SMN1; SMN2 Q16637 2/20 0.58
ATM Q13315 2/20 0.58
NPC1 O15118 1/20 0.58
CYP3A4 P08684 1/20 0.58
RAB9A P51151 1/20 0.58
KDM4E B2RXH2 2/20 0.56
HSD17B10 Q99714 2/20 0.56
IDO1 P14902 1/20 0.53
TDO2 P48775 1/20 0.53
NR1H4 Q96RI1 1/20 0.53
ESR1 P03372 1/20 0.53
SHBG P04278 1/20 0.53
ESR2 Q92731 1/20 0.53
LMNA P02545 3/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL235761 0.83 TTR (0.71) TTRALDH1A1MAPK1HPGDMEN1
SCHEMBL236891 0.82 TTR (0.70) TTRALDH1A1MEN1KMT2AATM
SCHEMBL232760 0.81 TTR (0.67) TTRALDH1A1MEN1KMT2AATM
SCHEMBL2330812 0.80 TTR (0.67) TTRALDH1A1MAPK1HPGDMEN1
SCHEMBL332837 0.80 TTR (0.66) TTRALDH1A1HPGDMEN1KMT2A
SCHEMBL5725941 0.79 L3MBTL1 (0.68) TTRALDH1A1MEN1KMT2ASMN1; SMN2
SCHEMBL1246697 0.78 RAB9A (0.65) TTRALDH1A1HPGDMEN1KMT2A
SCHEMBL29535974 0.77 MEN1 (0.70) TTRALDH1A1MAPK1HPGDMEN1
SCHEMBL1039742 0.77 SMN1; SMN2 (0.70) TTRALDH1A1MAPK1HPGDMEN1
SCHEMBL31511913 0.77 SMN1; SMN2 (0.70) TTRALDH1A1MAPK1HPGDMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 21 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230105307-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2023-04-06 US disclosed
US-11337935-B2 Identification of stabilizers of multimeric proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2022-05-24 US disclosed
US-20200016098-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2020-01-16 US disclosed
US-10278929-B2 Identification of stabilizers of multimeric proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2019-05-07 US disclosed
US-20190054040-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2019-02-21 US disclosed
US-10039726-B2 Identification of stabilizers of multimeric proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2018-08-07 US disclosed
US-10039726-B2 Identification of stabilizers of multimeric proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2018-08-07 US disclosed
EP-2346844-B1 SUBSTITUTED BENZFUROCHROMENES FOR THE PREVENTION AND TREATMENT OF BONE RELATED DISORDERS COUNCIL SCIENT IND RES (IN) 2017-09-20 EP disclosed
US-20160374961-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2016-12-29 US disclosed
US-9308209-B2 Identification of stabilizers of multimeric proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIO (US) 2016-04-12 US disclosed
US-20150126532-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2015-05-07 US disclosed
US-20150126532-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2015-05-07 US disclosed
US-8877795-B2 Identification of stabilizers of multimeric proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2014-11-04 US disclosed
US-8877795-B2 Identification of stabilizers of multimeric proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2014-11-04 US disclosed
US-20130203777-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2013-08-08 US disclosed
US-20130203777-A1 Identification of Stabilizers of Multimeric Proteins THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY 2013-08-08 US disclosed
US-20120003273-A1 SUBSTITUTED BENZFUROCHROMENES AND RELATED COMPOUNDS FOR THE PREVENTION AND TREATMENT OF BONE RELATED DISORDERS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (AN INDIAN REGISTERED BODY INCORPORATED UNDER THE REGISTRATION OF SOCIETIES ACT (ACT XXI OF 1860)) (IN) 2012-01-05 US disclosed
WO-2011140333-A1 IDENTIFICATION OF STABILIZERS OF MULTIMERIC PROTEINS THE BOARD OF TRUSTEES OF THE LELAND STANFORD JUNIOR UNIVERSITY (US) 2011-11-10 WO disclosed
EP-2346844-A1 SUBSTITUTED BENZFUROCHROMENES AND RELATED COMPOUNDS FOR THE PREVENTION AND TREATMENT OF BONE RELATED DISORDERS Council Of Scientific & Industrial Research (IN) 2011-07-27 EP disclosed
WO-2010052734-A1 SUBSTITUTED BENZFUROCHROMENES AND RELATED COMPOUNDS FOR THE PREVENTION AND TREATMENT OF BONE RELATED DISORDERS COUNCIL OF SCIENTIFIC & INDUSTRIAL RESEARCH (IN) 2010-05-14 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (10 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230105307-A1 Identification of Stabilizers of Multimeric Proteins TTR, HSPBP1, HSPH1 TTR 1/4885ALDH1A1 3493/4885MAPK1 4185/4885
US-20190054040-A1 Identification of Stabilizers of Multimeric Proteins TTR, HSPBP1, HSPH1 TTR 1/4885ALDH1A1 3493/4885MAPK1 4185/4885
US-10278929-B2 Identification of stabilizers of multimeric proteins TTR, HSPBP1, HSPH1 TTR 1/4885ALDH1A1 3296/4885MAPK1 4347/4885
US-11337935-B2 Identification of stabilizers of multimeric proteins TTR, HSPBP1, HSPH1 TTR 1/4885ALDH1A1 3493/4885MAPK1 4185/4885
US-20160374961-A1 Identification of Stabilizers of Multimeric Proteins TTR, ALB, HSPBP1 TTR 1/4885ALDH1A1 3246/4885MAPK1 4777/4885
US-10039726-B2 Identification of stabilizers of multimeric proteins TTR, ALB, HSPBP1 TTR 1/4885ALDH1A1 3246/4885MAPK1 4777/4885
US-20130203777-A1 Identification of Stabilizers of Multimeric Proteins TTR, HSPBP1, HSP90B1 TTR 1/4885ALDH1A1 3222/4885MAPK1 4663/4885
US-20150126532-A1 Identification of Stabilizers of Multimeric Proteins TTR, HSPBP1, HSPH1 TTR 1/4885ALDH1A1 3493/4885MAPK1 4185/4885
US-20200016098-A1 Identification of Stabilizers of Multimeric Proteins TTR, HSPBP1, HSPH1 TTR 1/4885ALDH1A1 3493/4885MAPK1 4185/4885
US-20120003273-A1 SUBSTITUTED BENZFUROCHROMENES AND RELATED COMPOUNDS FOR THE PREVENTION AND TREATMENT OF BONE RELATED DISORDERS AKR1C3, AKR1C4, SLC10A1 TTR 2235/4885ALDH1A1 1999/4885MAPK1 3299/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.