SCHEMBL23652001

SCHEMBL23652001

CNC(=O)Cc1cccc(OC(F)(F)F)c1

nearest known ligand 0.51

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
VNN1 O95497 1/20 0.51
GLS O94925 6/20 0.50
MAPK14 Q16539 1/20 0.50
P2RY14 Q15391 1/20 0.49
NLRP3 Q96P20 1/20 0.49
CHRM2 P08172 1/20 0.48
CHRM1 P11229 1/20 0.48
CHRM3 P20309 1/20 0.48
DGAT2 Q96PD7 1/20 0.48
FFAR2 O15552 1/20 0.47
BRAF P15056 1/20 0.47
CNR1 P21554 1/20 0.47
ROCK2 O75116 1/20 0.47
ROCK1 Q13464 1/20 0.47
NTRK1 P04629 1/20 0.47
MRGPRX4 Q96LA9 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21981021 0.87 AOC2 (0.51) VNN1GLSMAPK14P2RY14NLRP3
SCHEMBL378549 0.84 VNN1 (0.52) VNN1GLSMAPK14CHRM2CHRM1
SCHEMBL11546048 0.83 CHRM2 (0.51) VNN1GLSMAPK14CHRM2CHRM1
SCHEMBL28475012 0.83 VNN1 (0.56) VNN1GLSMAPK14CHRM2CHRM1
SCHEMBL13329837 0.81 NLRP3 (0.57) VNN1NLRP3
SCHEMBL10154070 0.81 POLB (0.60) GLS
SCHEMBL761677 0.81 MAPK14 (0.54) VNN1MAPK14CHRM2CHRM1CHRM3
SCHEMBL19914436 0.81 VNN1 (0.48) VNN1GLSMAPK14P2RY14FFAR2
SCHEMBL21484106 0.81 CTSD (0.45) VNN1GLSMAPK14P2RY14NLRP3
SCHEMBL21981003 0.80 GLS (0.49) VNN1GLSMAPK14P2RY14NLRP3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3954686-A1 HETEROCYCLIC GLUTAMINASE INHIBITORS Calithera Biosciences, Inc. (US) 2022-02-16 EP disclosed
EP-2920168-B1 HETEROCYCLIC GLUTAMINASE INHIBITORS CALITHERA BIOSCIENCES INC (US) 2021-07-21 EP disclosed