SCHEMBL2365727

SCHEMBL2365727

O=C(N[C@H]1C2CC3CC(C2)CC1(O)C3)c1cccc([S+]([O-])c2ccc(Cl)cn2)c1

nearest known ligand 0.37

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 1/20 0.37
HSD11B1 P28845 5/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
ALDH1A1 P00352 2/20 0.36
TSHR P16473 2/20 0.36
PKM P14618 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
SERPINE1 P05121 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
GRM5 P41594 4/20 0.33
FAAH O00519 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2369168 0.85 HSD11B1 (0.47) HSD11B1
SCHEMBL2365656 0.80 P2RX7 (0.39) P2RX7HSD11B1NPC1RAB9AALDH1A1
SCHEMBL2365755 0.79 PPARG (0.41) P2RX7NPC1PKMMEN1KMT2A
SCHEMBL2365635 0.74 IP6K1 (0.43) P2RX7HSD11B1NPC1TSHRSMN1; SMN2
SCHEMBL1675961 0.72 FAAH (0.55) P2RX7HSD11B1MEN1KMT2ATDP1
SCHEMBL2365642 0.68 FAAH (0.52) HSD11B1TDP1FAAHL3MBTL1
SCHEMBL2365627 0.65 IDH1 (0.57) HSD11B1MEN1KMT2A
SCHEMBL2365636 0.65 HSD11B1 (0.48) HSD11B1
SCHEMBL1168572 0.64 HSD11B1 (0.48) HSD11B1
SCHEMBL2365608 0.64 HSD11B1 (0.48) HSD11B1MEN1KMT2ATDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2362730-A1 ADAMANTYL BENZAMIDE COMPOUNDS High Point Pharmaceuticals, LLC (US) 2011-09-07 EP disclosed
WO-2010059618-A1 ADAMANTYL BENZAMIDE COMPOUNDS HIGH POINT PHARMACEUTICALS, LLC (US) 2010-05-27 WO disclosed