SCHEMBL23663156

SCHEMBL23663156

COc1ccc(Oc2c(Cl)cc(Br)cc2Cl)cc1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPBWR1 P48145 12/20 0.48
MCHR1 Q99705 4/20 0.43
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA7 P43166 1/20 0.42
CA9 Q16790 1/20 0.42
CA14 Q9ULX7 1/20 0.42
LTA4H P09960 2/20 0.42
SMN1; SMN2 Q16637 2/20 0.41
NPSR1 Q6W5P4 2/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 1/20 0.41
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 1/20 0.41
TAS1R3 Q7RTX0 1/20 0.41
TAS1R1 Q7RTX1 1/20 0.41
TAS1R2 Q8TE23 1/20 0.41
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17087154 0.86 NPBWR1 (0.52) NPBWR1MCHR1CA12CA1CA2
SCHEMBL3228597 0.81 TDP1 (0.50) NPBWR1MCHR1CA12CA1CA2
SCHEMBL29036495 0.80 THRB (0.35) NPBWR1MCHR1TAS1R3TAS1R1TAS1R2
SCHEMBL23663148 0.80 THRB (0.46) NPBWR1MCHR1CA12CA1CA2
Hydrochloric Acid SCHEMBL29965433 0.79 ALDH1A1 (0.52) NPBWR1MCHR1CA12CA1CA2
SCHEMBL23663189 0.79 NPBWR1 (0.43) NPBWR1MCHR1CA12CA1CA2
SCHEMBL23663172 0.78 TAS1R3 (0.45) NPBWR1MCHR1CA12CA1CA2
SCHEMBL11606863 0.78 MAPT (0.47) NPBWR1NPSR1LMNAMEN1ALDH1A1
SCHEMBL15713090 0.78 NPBWR1 (0.51) NPBWR1MCHR1MEN1KMT2ATHRA
SCHEMBL442742 0.77 ALDH1A1 (0.44) CA2ALDH1A1TAS1R3TAS1R1TAS1R2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20250320197-A1 THYROID HORMONE RECEPTOR AGONISTS AND USE THEREOF ECCOGENE INC (US) 2025-10-16 US disclosed
US-12291518-B2 Thyroid hormone receptor agonists and use thereof ECCOGENE INC. (US) 2025-05-06 US disclosed
CN-115244037-B Substituted triazinones as thyroid hormone receptor agonists 诚益生物(美国)公司 2024-10-25 CN disclosed
US-20240190846-A1 THYROID HORMONE RECEPTOR AGONISTS AND USE THEREOF ECCOGENE INC. 2024-06-13 US disclosed
US-11780825-B2 Thyroid hormone receptor agonists and use thereof ECCOGENE (SHANGHAI) CO., LTD. (CN) 2023-10-10 US disclosed
US-11780825-B2 Thyroid hormone receptor agonists and use thereof ECCOGENE (SHANGHAI) CO., LTD. (CN) 2023-10-10 US disclosed
US-11780825-B2 Thyroid hormone receptor agonists and use thereof ECCOGENE (SHANGHAI) CO., LTD. (CN) 2023-10-10 US disclosed
EP-4090652-A1 SUBSTITUTED TRIAZINONES AS THYROID HORMONE RECEPTOR AGONISTS Eccogene (Shanghai) Co., Ltd. (CN) 2022-11-23 EP disclosed
CN-115244037-A Substituted triazinones as thyroid hormone receptor agonists 上海诚益生物科技有限公司 2022-10-25 CN disclosed
US-20210230146-A1 THYROID HORMONE RECEPTOR AGONISTS AND USE THEREOF ECCOGENE INC. 2021-07-29 US disclosed
WO-2021143706-A1 SUBSTITUTED TRIAZINONES AS THYROID HORMONE RECEPTOR AGONISTS ECCOGENE (SHANGHAI) CO., LTD. (CN) 2021-07-22 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210230146-A1 THYROID HORMONE RECEPTOR AGONISTS AND USE THEREOF TSHR, THRA, THRB NPBWR1 154/4885MCHR1 56/4885CA12 1396/4885
US-11780825-B2 Thyroid hormone receptor agonists and use thereof TSHR, THRA, THRB NPBWR1 154/4885MCHR1 56/4885CA12 1396/4885
US-12291518-B2 Thyroid hormone receptor agonists and use thereof TSHR, THRA, THRB NPBWR1 154/4885MCHR1 56/4885CA12 1396/4885
US-20250320197-A1 THYROID HORMONE RECEPTOR AGONISTS AND USE THEREOF TSHR, THRA, THRB NPBWR1 154/4885MCHR1 56/4885CA12 1396/4885
US-20240190846-A1 THYROID HORMONE RECEPTOR AGONISTS AND USE THEREOF TSHR, THRA, THRB NPBWR1 154/4885MCHR1 56/4885CA12 1396/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.