SCHEMBL23673501

SCHEMBL23673501

O=C(O)C1(NC(c2ccoc2)C(F)(F)F)CCCCC1

nearest known ligand 0.37

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CTSK P43235 2/20 0.37
FAAH O00519 5/20 0.34
TRPV1 Q8NER1 3/20 0.34
USP2 O75604 1/20 0.32
HTT P42858 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
FABP4 P15090 1/20 0.32
FABP5 Q01469 1/20 0.32
CYP1A2 P05177 1/20 0.32
ERAP1 Q9NZ08 2/20 0.31
ALOX5 P09917 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4368196 0.82 CTSK (0.42) CTSKFAAHTRPV1FABP4FABP5
SCHEMBL13624184 0.81 CTSL (0.42) CTSKFABP4FABP5
SCHEMBL23693804 0.68 CTSK (0.33) CTSK
SCHEMBL1837046 0.67 KCNK3 (0.44) CTSKERAP1
SCHEMBL2156068 0.65 CTSK (0.66) CTSK
SCHEMBL5870313 0.63 ALDH1A1 (0.40) CTSKFAAHTRPV1USP2HTT
SCHEMBL8257823 0.63 ALDH1A1 (0.40) CTSKFAAHTRPV1USP2HTT
SCHEMBL12869545 0.61 ALDH1A1 (0.36) CTSKUSP2HTTSMN1; SMN2CYP1A2
SCHEMBL25152543 0.61 ALOX5 (0.33) ALOX5
SCHEMBL29154166 0.60 CYP1A2 (0.43) CTSKFAAHUSP2HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021147882-A1 DIBENZOFURAN DERIVATIVE CATHEPSIN K INHIBITOR, PREPARATION METHOD THEREFOR AND MEDICAL USE THEREOF 深圳信立泰药业股份有限公司 2021-07-29 WO disclosed