SCHEMBL2367383

SCHEMBL2367383

O=S(=O)(Nc1cccc2cc[nH]c12)c1ccccc1

nearest known ligand 0.71

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NR3C1 P04150 1/20 0.65
PGR P06401 1/20 0.65
NR3C2 P08235 1/20 0.65
AR P10275 1/20 0.65
RECQL P46063 1/20 0.59
ACLY P53396 1/20 0.53
SLC40A1 Q9NP59 4/20 0.52
ALDH1A1 P00352 3/20 0.52
AGTR1 P30556 2/20 0.52
GLO1 Q04760 2/20 0.52
PAX8 Q06710 2/20 0.52
G6PD P11413 1/20 0.52
NFKBIA P25963 1/20 0.52
METAP2 P50579 1/20 0.52
METAP1 P53582 1/20 0.52
ATM Q13315 1/20 0.52
TDP1 Q9NUW8 1/20 0.52
MEN1 O00255 1/20 0.52
MAPT P10636 1/20 0.52
KMT2A Q03164 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1984869 0.87 CA1 (0.60) NR3C1PGRNR3C2ARRECQL
SCHEMBL2367682 0.87 NR3C1 (0.64) NR3C1PGRNR3C2ARSLC40A1
SCHEMBL2367735 0.87 NR3C1 (0.60) NR3C1PGRNR3C2ARACLY
SCHEMBL3061760 0.86 NR3C1 (0.56) NR3C1PGRNR3C2ARRECQL
SCHEMBL3066019 0.84 SLC40A1 (0.57) NR3C1PGRNR3C2ARACLY
SCHEMBL2367583 0.83 NFKBIA (0.58) NR3C1PGRNR3C2ARNFKBIA
SCHEMBL2403697 0.83 TUBB4A (0.61) NR3C1PGRNR3C2ARSLC40A1
SCHEMBL3073814 0.83 NR3C1 (0.56) NR3C1PGRNR3C2ARRECQL
SCHEMBL3061022 0.83 GLO1 (0.58) NR3C1PGRNR3C2ARACLY
SCHEMBL1207409 0.83 SLC40A1 (0.62) NR3C1PGRNR3C2ARSLC40A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 11 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2366687-B1 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO LTD (CN) 2015-11-04 EP disclosed
EP-1644367-B1 IMMUNOSUPPRESSANT COMPOUNDS AND COMPOSITIONS NOVARTIS AG (CH) 2015-10-14 EP disclosed
US-8173693-B2 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO., LTD. (TW) 2012-05-08 US disclosed
US-8173693-B2 Benzenesulfonamide derivatives and pharmaceutical composition thereof PURZER PHARMACEUTICAL CO., LTD. (TW) 2012-05-08 US disclosed
CN-102199148-A Benzenesulfonamide derivatives and pharmaceutical compositions thereof PURZER PHARMACEUTICAL CO LTD 2011-09-28 CN disclosed
US-20110230651-A1 Benzenesulfonamide derivatives and pharmaceutical composition therof PURZER PHARMACEUTICAL CO., LTD. (TW) 2011-09-22 US disclosed
US-20110230651-A1 Benzenesulfonamide derivatives and pharmaceutical composition therof PURZER PHARMACEUTICAL CO., LTD. (TW) 2011-09-22 US disclosed
EP-2366687-A2 Benzenesulfonamide derivatives and pharmaceutical composition thereof Purzer Pharmaceutical Co., Ltd. (CN) 2011-09-21 EP disclosed
CN-100356979-C Integrin expression inhibitors EISAI CO LTD (JP) 2007-12-26 CN disclosed
EP-1783496-A1 METHOD OF ANALYZING PROTEIN STRUCTURAL AFFINITY RELATIONSHIP Eisai R&D Management Co., Ltd. (JP) 2007-05-09 EP disclosed
CN-1396833-A Integrin expression inhibitors EISAI CO LTD (JP) 2003-02-12 CN disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110230651-A1 Benzenesulfonamide derivatives and pharmaceutical composition therof CCNI, CCNE1, CCND1 NR3C1 4137/4885PGR 1644/4885NR3C2 4025/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.