SCHEMBL2368752

SCHEMBL2368752

COc1cccc(-c2csc3ncncc23)c1

nearest known ligand 0.53

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PKM P14618 1/20 0.53
CYP2C19 P33261 12/20 0.52
CYP1A2 P05177 11/20 0.52
CYP3A4 P08684 11/20 0.52
CYP2D6 P10635 11/20 0.52
HSD17B10 Q99714 8/20 0.52
MAPK1 P28482 5/20 0.52
LMNA P02545 8/20 0.51
CLK4 Q9HAZ1 8/20 0.51
ALDH1A1 P00352 7/20 0.51
CYP2C9 P11712 5/20 0.51
TSHR P16473 5/20 0.51
ALOX15 P16050 4/20 0.51
MAPT P10636 4/20 0.50
HPGD P15428 2/20 0.50
KDM4E B2RXH2 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
MITF O75030 1/20 0.49
HTT P42858 1/20 0.49
PIP4K2C Q8TBX8 1/20 0.49

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14964882 0.78 FGFR1 (0.53) CYP2C19CYP1A2MAPK1LMNACLK4
SCHEMBL2368453 0.76 PKM (0.51) PKMCYP2C19CYP1A2CYP3A4CYP2D6
SCHEMBL2369304 0.75 CYP2A6 (0.51) MAPK1MAPT
SCHEMBL2367997 0.74 LMNA (0.49) PKMLMNACLK4ALDH1A1MAPT
SCHEMBL16294249 0.73 CYP3A4 (0.54) CYP2C19CYP1A2CYP3A4CYP2D6HSD17B10
SCHEMBL5376619 0.73 MAPT (0.53) MAPK1LMNAALDH1A1MAPTHPGD
SCHEMBL2368915 0.71 SMN1; SMN2 (0.38) CYP2C19CYP1A2CYP3A4HSD17B10MAPK1
SCHEMBL30700550 0.71 DHFR (0.41) LMNACLK4ALDH1A1MAPTKDM4E
SCHEMBL12599829 0.71 PKM (0.60) PKMHSD17B10MAPK1LMNACLK4
SCHEMBL12303147 0.71 DYRK1A (0.55) CYP2C19CYP1A2CYP3A4CYP2D6HSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8022076-B2 Thieno[2,3-d]pyrimidine derivatives as potassium channel modulators; antiarrhythmia agents XENTION LIMITED (GB) 2011-09-20 US disclosed