SCHEMBL23715829

SCHEMBL23715829

N=C(NC(=O)c1ccccc1)C(NNOc1cccc(Cl)c1)c1ccccc1

nearest known ligand 0.44

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
S1PR3 Q99500 15/20 0.44
S1PR1 P21453 5/20 0.44
S1PR4 O95977 5/20 0.43
S1PR5 Q9H228 1/20 0.43
NPC1 O15118 2/20 0.40
RAB9A P51151 2/20 0.40
S1PR2 O95136 2/20 0.40
KCNK3 O14649 1/20 0.39
KCNK9 Q9NPC2 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23715916 0.81 OGG1 (0.44) CYP1A2CYP2D6CYP2C9CYP2C19
SCHEMBL23715832 0.81 S1PR3 (0.58) S1PR3S1PR1S1PR4S1PR5S1PR2
SCHEMBL17664156 0.79 S1PR3 (0.61) S1PR3S1PR1S1PR4S1PR5S1PR2
SCHEMBL23715936 0.79 NPC1 (0.44) NPC1RAB9ACYP1A2CYP2D6CYP2C9
SCHEMBL23716312 0.77 S1PR3 (0.52) S1PR3S1PR1S1PR4S1PR5S1PR2
SCHEMBL21130417 0.77 S1PR3 (0.50) S1PR3S1PR1S1PR4S1PR5NPC1
SCHEMBL23716111 0.74 OGG1 (0.45)
SCHEMBL23716193 0.73 OGG1 (0.44)
SCHEMBL23716102 0.72 S1PR3 (0.40) S1PR3S1PR1S1PR4S1PR5S1PR2
SCHEMBL23715998 0.71 S1PR3 (0.42) S1PR3S1PR1S1PR4S1PR5S1PR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3209732-B1 SPHINGOSINE-1-PHOSPATE RECEPTOR MODULATORS FOR TREATMENT OF CARDIOPULMONARY DISORDERS SCRIPPS RESEARCH INST (US) 2021-08-04 EP disclosed