SCHEMBL23770634

SCHEMBL23770634

Cc1ccccc1-c1nc(N[S+]([O-])c2cccc(N3CCCC(F)CNCC3)n2)ccc1C(F)(F)F

nearest known ligand 0.34

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
CYP1A2 P05177 3/20 0.34
CYP2C9 P11712 1/20 0.34
CCNT1 O60563 3/20 0.33
CCNK O75909 3/20 0.33
CCNE1 P24864 3/20 0.33
CDK2 P24941 3/20 0.33
CDK9 P50750 3/20 0.33
CDK12 Q9NYV4 3/20 0.33
ADRB2 P07550 1/20 0.32
CYP2C19 P33261 1/20 0.31
SOS1 Q07889 3/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770787 0.87 PDE10A (0.35) CYP1A2CYP2C9CYP2C19
SCHEMBL23770621 0.86 PDE10A (0.35) CYP1A2CYP2C9CYP2C19
SCHEMBL23770649 0.82 PIM1 (0.34) CYP1A2
SCHEMBL23770643 0.80 ADRB2 (0.37) CYP1A2CYP2C9ADRB2CYP2C19SOS1
SCHEMBL23770598 0.80 ADRB2 (0.43) CYP1A2CYP2C9ADRB2CYP2C19
SCHEMBL23770766 0.80 PRKCQ (0.35) CYP1A2CYP2C9
SCHEMBL23770416 0.80 PTPN11 (0.37)
SCHEMBL23770413 0.78 CCNT1 (0.47) CCNT1CCNKCCNE1CDK2CDK9
SCHEMBL23770712 0.78 NPC1 (0.33) CYP1A2CYP2C19
SCHEMBL23770480 0.77 GRIN2B (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed