SCHEMBL23770840

SCHEMBL23770840

Cc1ccccc1-c1nc(NSc2cccc(N3CCC(C)CC3)n2)ccc1C(F)(F)F

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 4/20 0.35
ALDH1A1 P00352 4/20 0.35
MAPT P10636 2/20 0.35
TDP1 Q9NUW8 2/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
MAPK13 O15264 1/20 0.33
MAPK12 P53778 1/20 0.33
MAPK11 Q15759 1/20 0.33
MAPK14 Q16539 1/20 0.33
AR P10275 1/20 0.33
TSHR P16473 2/20 0.32
CYP1A2 P05177 2/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C19 P33261 1/20 0.32
HSD17B10 Q99714 1/20 0.32
HPGD P15428 1/20 0.32
LMNA P02545 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23770725 0.92 CYP1A2 (0.37) KDM4EALDH1A1TDP1MEN1KMT2A
SCHEMBL23770433 0.91 PDE10A (0.36) KDM4EALDH1A1TDP1L3MBTL1MEN1
SCHEMBL23770664 0.90 NPY5R (0.36) KDM4EALDH1A1TDP1L3MBTL1MEN1
SCHEMBL23770859 0.89 CYP1A2 (0.44) KDM4EALDH1A1TDP1TSHRCYP1A2
SCHEMBL23770653 0.88 CNR2 (0.40) ALDH1A1MAPTTSHRCYP1A2CYP3A4
SCHEMBL23770663 0.88 CYP1A2 (0.43) KDM4EALDH1A1TDP1MEN1KMT2A
SCHEMBL23770673 0.88 HRH4 (0.35)
SCHEMBL23770658 0.86 CTSS (0.31)
SCHEMBL23770753 0.86 GRIN2B (0.36) GRIN2B
SCHEMBL23770647 0.86 KDM4E (0.33) KDM4EALDH1A1TDP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3504194-B1 N-(PYRIDIN-2-YL)PYRIDINE-SULFONAMIDE DERIVATIVES AND THEIR USE IN THE TREATMENT OF DISEASE NOVARTIS AG (CH) 2021-08-18 EP disclosed