SCHEMBL23809138

SCHEMBL23809138

Cc1nc(CN2CCC(O)C2)nc(C)c1C(C)(C)C

nearest known ligand 0.40

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
GAA P10253 2/20 0.40
KDM4E B2RXH2 1/20 0.40
XBP1 P17861 1/20 0.40
MAPK1 P28482 1/20 0.40
HTT P42858 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
CD274 Q9NZQ7 6/20 0.38
PDCD1LG2 Q9BQ51 3/20 0.38
SYK P43405 3/20 0.35
PDCD1 Q15116 3/20 0.35
PDE2A O00408 1/20 0.34
PDE5A O76074 1/20 0.34
PDE11A Q9HCR9 1/20 0.34
PDE10A Q9Y233 1/20 0.34
CNR2 P34972 3/20 0.33
CYP3A4 P08684 1/20 0.33
JAK3 P52333 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL26580970 0.84 CD274 (0.43) ALDH1A1GAAKDM4EXBP1MAPK1
SCHEMBL26038021 0.79 CD274 (0.38) ALDH1A1CD274PDCD1LG2SYKPDCD1
SCHEMBL23809141 0.76 SIGMAR1 (0.46) ALDH1A1KDM4EMAPK1HTT
SCHEMBL23808976 0.73 ALDH1A1 (0.41) ALDH1A1GAAKDM4EHTT
SCHEMBL23809104 0.72 NPSR1 (0.38) ALDH1A1KDM4EHTTNPSR1
SCHEMBL23809108 0.72 CXCR4 (0.39) ALDH1A1KDM4EHTT
SCHEMBL23809035 0.72 ALOX15 (0.43) ALDH1A1GAAKDM4EHTTCNR2
SCHEMBL23809134 0.71 HRH3 (0.44) ALDH1A1CD274PDCD1LG2
SCHEMBL31662619 0.68 ALDH1A1 (0.57) ALDH1A1GAAKDM4EXBP1MAPK1
SCHEMBL23809110 0.68 LMNA (0.37) ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20210283138-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS VANDERBILT UNIVERSITY 2021-09-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210283138-A1 SUBSTITUTED INDOLE MCL-1 INHIBITORS MCL1, BCL2L1, BCL9 ALDH1A1 2556/4885GAA 3420/4885KDM4E 1156/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.