SCHEMBL23901369

SCHEMBL23901369

OC(c1cc(F)cc(F)c1)c1ccc2[nH]ncc2c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.45
GRIN2B Q13224 2/20 0.45
CTNNB1 P35222 1/20 0.45
WNT3A P56704 1/20 0.45
MAOB P27338 1/20 0.44
NOS1 P29475 3/20 0.44
RAB9A P51151 3/20 0.44
ROCK1 Q13464 3/20 0.44
CSNK2A1 P68400 2/20 0.44
METAP2 P50579 1/20 0.44
KDM4E B2RXH2 1/20 0.44
MEN1 O00255 1/20 0.44
ALDH1A1 P00352 1/20 0.44
GAA P10253 1/20 0.44
MAPT P10636 1/20 0.44
HPGD P15428 1/20 0.44
KMT2A Q03164 1/20 0.44
HIF1A Q16665 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
NPC1 O15118 2/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1363970 0.81 DYRK3 (0.54) ROCK2GRIN2BCTNNB1WNT3ANOS1
SCHEMBL3497213 0.76 TRPA1 (0.59) ROCK2CTNNB1WNT3AMAOBNOS1
SCHEMBL30074251 0.76 ROCK2 (0.50) ROCK2GRIN2BCTNNB1WNT3AMAOB
SCHEMBL29520764 0.75 TRPA1 (0.54) ROCK2MAOBNOS1RAB9AROCK1
SCHEMBL27771848 0.75 GRIN2B (0.49) ROCK2GRIN2BCTNNB1WNT3AMAOB
SCHEMBL12181364 0.75 NOS1 (0.46) ROCK2GRIN2BCTNNB1WNT3AMAOB
SCHEMBL28999426 0.72 GSK3B (0.64) ROCK2MAOBNOS1RAB9AROCK1
SCHEMBL27750996 0.72 NOS1 (0.50) ROCK2GRIN2BCTNNB1WNT3AMAOB
SCHEMBL84462 0.72 TRPA1 (0.54) ROCK2MAOBNOS1RAB9AROCK1
SCHEMBL30141452 0.71 ROCK2 (0.42) ROCK2CTNNB1WNT3AMAOBNOS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115916771-A Multi-target antitumor compound and preparation method and application thereof 浙江华海药业股份有限公司 2023-04-04 CN disclosed
WO-2021197467-A1 MULTI-TARGET ANTI-TUMOR COMPOUND, PREPARATION METHOD THEREFOR AND USE THEREOF 上海华汇拓医药科技有限公司 2021-10-07 WO disclosed