SCHEMBL23907993

SCHEMBL23907993

CSc1ncc(F)c(OCC(=O)NC2C3CC4CC(C3)CC2C4)n1

nearest known ligand 0.45

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRB P10828 4/20 0.45
L3MBTL1 Q9Y468 1/20 0.39
HSD11B1 P28845 4/20 0.38
EPHX2 P34913 5/20 0.36
LMNA P02545 2/20 0.34
HTT P42858 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23907995 0.80 ALDH1A1 (0.47) THRBL3MBTL1LMNAHTT
SCHEMBL23900450 0.76 THRB (0.42) THRBL3MBTL1HSD11B1EPHX2
SCHEMBL23907980 0.68 ALDH1A1 (0.51) THRBLMNAHTT
SCHEMBL23907985 0.67 ALDH1A1 (0.47) THRBL3MBTL1LMNAHTT
SCHEMBL4404236 0.66 EPHX2 (0.52) THRBHSD11B1EPHX2
SCHEMBL3456922 0.65 MEN1 (0.61) L3MBTL1HSD11B1LMNAHTT
SCHEMBL23900434 0.65 THRB (0.44) THRBL3MBTL1HSD11B1EPHX2LMNA
SCHEMBL4784023 0.64 RAB9A (0.66) LMNAHTT
SCHEMBL23884322 0.63 ALDH1A1 (0.43) THRBL3MBTL1LMNAHTT
SCHEMBL11353062 0.60 HSD11B1 (0.55) THRBL3MBTL1HSD11B1EPHX2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240182450-A1 Novel 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses OREGON HEALTH AND SCIENCE UNIVERSITY 2024-06-06 US disclosed
US-11932626-B2 2-pyrimidone analogs as potent antiviral agents against Alphaviruses SOUTHERN RESEARCH INSTITUTE (US) 2024-03-19 US disclosed
US-20230120566-A1 Novel 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses OREGON HEALTH AND SCIENCE UNIVERSITY 2023-04-20 US disclosed
CN-115916175-A Novel 2-pyrimidinone analogs as potent antiviral agents against alphaviruses 南方研究院 2023-04-04 CN disclosed
US-11566019-B2 2-pyrimidone analogs as potent antiviral agents against alphaviruses SOUTHERN RESEARCH INSTITUTE (US) 2023-01-31 US disclosed
US-20220177452-A9 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2022-06-09 US disclosed
US-20210317106-A1 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses SOUTHERN RES INST (US) 2021-10-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (6 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210317106-A1 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses EIF2AK2, ZC3HAV1, MAVS THRB 3748/4885L3MBTL1 390/4885HSD11B1 4069/4885
US-11566019-B2 2-pyrimidone analogs as potent antiviral agents against alphaviruses EIF2AK2, ZC3HAV1, MAVS THRB 3748/4885L3MBTL1 390/4885HSD11B1 4069/4885
US-11932626-B2 2-pyrimidone analogs as potent antiviral agents against Alphaviruses EIF2AK2, ZC3HAV1, MAVS THRB 3748/4885L3MBTL1 390/4885HSD11B1 4069/4885
US-20220177452-A9 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses EIF2AK2, ZC3HAV1, MAVS THRB 3748/4885L3MBTL1 390/4885HSD11B1 4069/4885
US-20240182450-A1 Novel 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses EIF2AK2, ZC3HAV1, MAVS THRB 3761/4885L3MBTL1 450/4885HSD11B1 3980/4885
US-20230120566-A1 Novel 2-Pyrimidone Analogs as Potent Antiviral Agents Against Alphaviruses EIF2AK2, ZC3HAV1, MAVS THRB 3761/4885L3MBTL1 450/4885HSD11B1 3980/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.