SCHEMBL2391401

SCHEMBL2391401

O=C(O)C1(NCc2ccccc2)COC1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LTA4H P09960 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.41
EPHX1 P07099 2/20 0.41
USP2 O75604 1/20 0.41
HTT P42858 1/20 0.41
LMNA P02545 2/20 0.41
CFD P00746 1/20 0.41
GSK3B P49841 2/20 0.40
BCHE P06276 1/20 0.40
TP53 P04637 1/20 0.40
KDM4E B2RXH2 2/20 0.40
GAA P10253 2/20 0.40
ALDH1A1 P00352 1/20 0.40
HSP90AA1 P07900 1/20 0.40
HSP90AB1 P08238 1/20 0.40
MAPT P10636 1/20 0.40
APEX1 P27695 1/20 0.40
RECQL P46063 1/20 0.40
HSD17B10 Q99714 1/20 0.40
TDP1 Q9NUW8 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10458177 0.84 LTA4H (0.51) LTA4HSMN1; SMN2EPHX1USP2TP53
SCHEMBL15221427 0.84 LTA4H (0.50) LTA4HSMN1; SMN2EPHX1USP2HTT
SCHEMBL5320356 0.81 LTA4H (0.59) LTA4HSMN1; SMN2EPHX1USP2LMNA
Hydrochloric Acid SCHEMBL6008696 0.79 LTA4H (0.57) LTA4HSMN1; SMN2EPHX1USP2LMNA
SCHEMBL5678125 0.79 LTA4H (0.57) LTA4HSMN1; SMN2EPHX1USP2LMNA
SCHEMBL29131629 0.77 CFD (0.42) SMN1; SMN2EPHX1USP2HTTLMNA
SCHEMBL31310044 0.75 IDO1 (0.38) EPHX1USP2HTTLMNACFD
SCHEMBL12873787 0.74 LTA4H (0.42) LTA4HSMN1; SMN2EPHX1USP2HTT
SCHEMBL17459841 0.74 IDO1 (0.41) USP2HTTCFDKDM4EGAA
SCHEMBL30362851 0.74 SMN1; SMN2 (0.46) SMN1; SMN2EPHX1TP53KDM4EGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20240300965-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2024-09-12 US disclosed
US-11999746-B2 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2024-06-04 US disclosed
US-20200055863-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-02-20 US disclosed
US-20200055863-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2020-02-20 US disclosed
US-10428078-B2 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-10-01 US disclosed
US-10428078-B2 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-10-01 US disclosed
EP-3172211-B1 TRICYCLIC IMIDAZO-PYRIMIDINONE DERIVATIVES FOR THE TREATMENT OF DISEASES MEDIATED BY LP-PLA2 GLAXOSMITHKLINE IP DEV LTD (GB) 2019-07-03 EP disclosed
EP-3172211-B1 TRICYCLIC IMIDAZO-PYRIMIDINONE DERIVATIVES FOR THE TREATMENT OF DISEASES MEDIATED BY LP-PLA2 GLAXOSMITHKLINE IP DEV LTD (GB) 2019-07-03 EP disclosed
US-20190023715-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-01-24 US disclosed
US-20190023715-A1 COMPOUNDS GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2019-01-24 US disclosed
US-10125141-B2 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2018-11-13 US disclosed
US-20170204109-A1 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-07-20 US disclosed
US-20170204109-A1 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-07-20 US disclosed
US-20170204109-A1 Compounds GLAXOSMITHKLINE INTELLECTUAL PROPERTY DEVELOPMENT LIMITED (GB) 2017-07-20 US disclosed
US-20110224188-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-alpha]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-09-15 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224188-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-alpha]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES HPGDS, COL14A1, ARG1 LTA4H 612/4885SMN1; SMN2 3828/4885EPHX1 3366/4885
US-20200055863-A1 COMPOUNDS PLAAT2, PLA2G12A, PLA2G1B LTA4H 36/4885SMN1; SMN2 1367/4885EPHX1 196/4885
US-20190023715-A1 COMPOUNDS PLAAT2, PLA2G12A, PLA2G1B LTA4H 36/4885SMN1; SMN2 1367/4885EPHX1 196/4885
US-10125141-B2 Compounds PLAAT2, PLA2G12A, PLA2G1B LTA4H 36/4885SMN1; SMN2 1367/4885EPHX1 196/4885
US-10428078-B2 Compounds PLAAT2, PLA2G12A, PLA2G1B LTA4H 36/4885SMN1; SMN2 1367/4885EPHX1 196/4885
US-20240300965-A1 COMPOUNDS PLAAT2, PLA2G12A, PLA2G1B LTA4H 36/4885SMN1; SMN2 1367/4885EPHX1 196/4885
US-11999746-B2 Compounds PLAAT2, PLA2G12A, PLA2G1B LTA4H 36/4885SMN1; SMN2 1367/4885EPHX1 196/4885
US-20170204109-A1 Compounds PLAAT2, PLA2G12A, PLA2G1B LTA4H 36/4885SMN1; SMN2 1367/4885EPHX1 196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.