SCHEMBL23928418

SCHEMBL23928418

Cc1nn(C(F)F)cc1NC(N)=O

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.37
ALDH1A1 P00352 1/20 0.37
LRRK2 Q5S007 2/20 0.36
RORC P51449 1/20 0.34
CYP2C9 P11712 2/20 0.33
CYP2B6 P20813 2/20 0.33
CYP2C19 P33261 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP1A2 P05177 1/20 0.32
CYP2C8 P10632 1/20 0.32
CYP2D6 P10635 1/20 0.32
POLB P06746 2/20 0.32
CDK8 P49336 1/20 0.31
ATM Q13315 1/20 0.31
KIF11 P52732 1/20 0.31
KDM4E B2RXH2 1/20 0.31
GAA P10253 1/20 0.31
ITK Q08881 1/20 0.31
BACE1 P56817 1/20 0.31
BACE2 Q9Y5Z0 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21246184 0.76 LMNA (0.56) LMNAALDH1A1CYP2C9CYP2C19CYP1A2
SCHEMBL24707430 0.71 LRRK2 (0.36) LRRK2RORCBACE1
SCHEMBL22637868 0.69 ALKBH1 (0.36) ALDH1A1POLBKDM4E
SCHEMBL26425463 0.69 GAA (0.43) ALDH1A1CYP2C9CYP2C19CYP1A2POLB
SCHEMBL18898579 0.67 LRRK2 (0.33) LRRK2
Hydrochloric Acid SCHEMBL26643669 0.66
SCHEMBL22013691 0.65 LRRK2 (0.34) LRRK2
SCHEMBL24753795 0.65 LRRK2 (0.37) LRRK2
SCHEMBL16679625 0.64 BRD4 (0.30)
SCHEMBL12272890 0.64 ADCY10 (0.35) LRRK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11230545-B2 Heterocyclic compound TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2022-01-25 US disclosed
US-20210332045-A1 HETEROCYCLIC COMPOUND TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2021-10-28 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11230545-B2 Heterocyclic compound MALT1, SQSTM1, PPM1D LMNA 3838/4885ALDH1A1 1199/4885LRRK2 2080/4885
US-20210332045-A1 HETEROCYCLIC COMPOUND MALT1, SQSTM1, PPM1D LMNA 3838/4885ALDH1A1 1199/4885LRRK2 2080/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.