SCHEMBL26425463

SCHEMBL26425463

CNC(=O)c1cn(C(F)F)nc1C

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
GAA P10253 7/20 0.43
BAZ2B Q9UIF8 1/20 0.40
ATM Q13315 1/20 0.35
ALDH1A1 P00352 3/20 0.34
CYP1A2 P05177 2/20 0.34
CYP2C9 P11712 2/20 0.34
NAMPT P43490 2/20 0.34
BRD4 O60885 2/20 0.33
RAB9A P51151 2/20 0.33
ALPL P05186 1/20 0.33
CYP2C19 P33261 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
MAPK1 P28482 1/20 0.32
NPC1 O15118 1/20 0.32
MAPT P10636 1/20 0.32
POLB P06746 1/20 0.31
ALK Q9UM73 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22637868 0.81 ALKBH1 (0.36) ALDH1A1MAPTPOLB
SCHEMBL8568083 0.75 GAA (0.69) GAABAZ2BATMALDH1A1CYP1A2
SCHEMBL20028548 0.74 TSHR (0.43) BAZ2BALDH1A1RAB9ANPC1MAPT
SCHEMBL17741451 0.72 BACE1 (0.42) RAB9A
SCHEMBL22979652 0.70 P2RX7 (0.42) GAAATMALDH1A1CYP1A2CYP2C9
SCHEMBL23928418 0.69 LMNA (0.37) GAAATMALDH1A1CYP1A2CYP2C9
SCHEMBL13975783 0.68 BAZ2B (0.45) BAZ2BBRD4
SCHEMBL30147529 0.67 PLK1 (0.43) SMN1; SMN2
SCHEMBL30147538 0.67 PLK1 (0.49) SMN1; SMN2
SCHEMBL12092481 0.67 GAA (0.43) GAABAZ2BALDH1A1CYP1A2CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2023192901-A9 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-12-14 WO disclosed
WO-2023192901-A1 QUINOLINE DERIVATIVES AS MODULATORS OF MAS-RELATED G-PROTEIN RECEPTOR X2 AND RELATED PRODUCTS ESCIENT PHARMACEUTICALS, INC. (US) 2023-10-05 WO disclosed