SCHEMBL23937727

SCHEMBL23937727

CCCC(=O)c1cnc(N)n1CC

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.33
KMT2A Q03164 2/20 0.33
HPGD P15428 3/20 0.33
ALDH1A1 P00352 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
RECQL P46063 1/20 0.33
HSD17B10 Q99714 1/20 0.33
TDP1 Q9NUW8 1/20 0.33
CYP1A2 P05177 2/20 0.32
F2 P00734 1/20 0.32
CYP2C19 P33261 1/20 0.32
GABRA1 P14867 2/20 0.32
GABRG2 P18507 2/20 0.32
GABRB3 P28472 2/20 0.32
GABRA5 P31644 2/20 0.32
GABRA3 P34903 2/20 0.32
GABRA2 P47869 2/20 0.32
EEF2K O00418 1/20 0.32
GABRP O00591 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10235408 0.65 CYP1A2 (0.36) KMT2AALDH1A1ALOX15TDP1CYP1A2
SCHEMBL21393806 0.65 NOS3 (0.40) HPGDALDH1A1TSHRHSD17B10CYP1A2
SCHEMBL13838594 0.62 SMN1; SMN2 (0.56) HSD17B3HPGDGABRA1GABRG2GABRB3
SCHEMBL10183000 0.62 CYP1A2 (0.38) KMT2AALDH1A1ALOX15TDP1CYP1A2
SCHEMBL3551145 0.61 ALOX15 (0.43) ALDH1A1ALOX15SMN1; SMN2
SCHEMBL6106298 0.61 MAPK1 (0.40) KMT2AALDH1A1TSHRSMN1; SMN2L3MBTL1
SCHEMBL1979899 0.60 CSNK1D (0.49) KMT2AHPGDALDH1A1HSD17B10CYP1A2
SCHEMBL1752323 0.60 GPR35 (0.40) KMT2AHPGDALDH1A1ALOX15TSHR
SCHEMBL17819955 0.60 GABRA1 (0.47) HSD17B3KMT2AHPGDALDH1A1ALOX15
SCHEMBL2281613 0.60 MAPK1 (0.33) KMT2AALDH1A1ALOX15TSHRTDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed