SCHEMBL23937731

SCHEMBL23937731

CCc1cc2ccn(C)c2nn1

nearest known ligand 0.33

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
PIK3CB P42338 1/20 0.33
PRKCI P41743 1/20 0.32
APP P05067 1/20 0.31
KDM1A O60341 1/20 0.31
HSD11B1 P28845 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23937734 0.86 NOS3 (0.33) PIK3CBPRKCI
SCHEMBL23937732 0.76 CYP11B1 (0.36)
SCHEMBL13514036 0.73 DDB1 (0.37) PIK3CB
SCHEMBL20674183 0.73 PIK3CB (0.34) PIK3CBPRKCIAPPHSD11B1
SCHEMBL23937882 0.69 GRM1 (0.36) PIK3CB
SCHEMBL20631760 0.69 XDH (0.35) PIK3CBPRKCIKDM1A
SCHEMBL12524710 0.69 CHRNA7 (0.41) PIK3CBAPP
SCHEMBL13824599 0.66
SCHEMBL21281472 0.66 PIK3CB (0.46) PIK3CBPRKCIKDM1AHSD11B1
SCHEMBL23937773 0.66 BRD9 (0.33) PIK3CBAPP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed