SCHEMBL23937859

SCHEMBL23937859

CCOc1cnc(CC)nc1O

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AOC3 Q16853 2/20 0.36
ALDH1A1 P00352 2/20 0.32
KDM4E B2RXH2 1/20 0.32
MAPK1 P28482 1/20 0.32
HSD17B10 Q99714 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
FOS P01100 2/20 0.32
JUN P05412 2/20 0.32
NFKB1 P19838 2/20 0.32
NFKB2 Q00653 2/20 0.32
RELA Q04206 2/20 0.32
SMN1; SMN2 Q16637 2/20 0.31
LMNA P02545 1/20 0.31
TLR8 Q9NR97 1/20 0.31
HCRTR1 O43613 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
MAPT P10636 2/20 0.31
L3MBTL1 Q9Y468 2/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL11524601 0.85 HTT (0.34) ALDH1A1KDM4EHSD17B10LMNATLR8
SCHEMBL11790398 0.82 AOC3 (0.37) AOC3ALDH1A1KDM4EMAPK1HSD17B10
SCHEMBL11202958 0.81 AOC3 (0.32) AOC3
SCHEMBL2148346 0.80 AOC3 (0.38) AOC3ALDH1A1KDM4EMAPK1HSD17B10
SCHEMBL2876075 0.76 ALOX15 (0.41) ALDH1A1SMN1; SMN2LMNAL3MBTL1
SCHEMBL13727051 0.75 LMNA (0.30) TSHRLMNA
SCHEMBL10689547 0.74 AOC3 (0.34) AOC3ALDH1A1KDM4EMAPK1HSD17B10
SCHEMBL7606690 0.74 NOS3 (0.31) FOSJUNNFKB1NFKB2RELA
SCHEMBL10998377 0.72 DHFR (0.33)
SCHEMBL15196099 0.72 TSHR (0.30) TSHRSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3399968-B1 SELECTIVE INHIBITORS OF CLINICALLY IMPORTANT MUTANTS OF THE EGFR TYROSINE KINASE CS PHARMATECH LTD (KY) 2021-10-20 EP disclosed