SCHEMBL2393997

SCHEMBL2393997

NC(=O)c1ncccc1C=O

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRIM24 O15164 2/20 0.50
TRIM33 Q9UPN9 2/20 0.50
KDM4E B2RXH2 4/20 0.42
KMT2A Q03164 3/20 0.42
NPSR1 Q6W5P4 2/20 0.42
L3MBTL1 Q9Y468 2/20 0.42
MEN1 O00255 2/20 0.42
NPC1 O15118 1/20 0.42
HSP90AA1 P07900 1/20 0.42
IDO1 P14902 1/20 0.42
RAB9A P51151 1/20 0.42
BLM P54132 2/20 0.41
MAPT P10636 2/20 0.41
ALDH1A1 P00352 1/20 0.41
CYP3A4 P08684 1/20 0.41
ALOX15 P16050 1/20 0.41
TSHR P16473 1/20 0.41
AGER Q15109 1/20 0.41
F7 P08709 1/20 0.41
F3 P13726 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7222788 0.83 KDM4E (0.40) TRIM24TRIM33KDM4ENPSR1L3MBTL1
SCHEMBL2840909 0.83 KDM4E (0.40) TRIM24TRIM33KDM4ENPSR1L3MBTL1
SCHEMBL547926 0.82 KDM4E (0.57) TRIM24TRIM33KDM4EKMT2ANPSR1
SCHEMBL29950595 0.81 TRIM24 (0.50) TRIM24TRIM33KDM4EKMT2ANPSR1
SCHEMBL1515655 0.80 MKNK1 (0.38) TRIM24TRIM33KDM4ENPSR1L3MBTL1
SCHEMBL14152216 0.79 NFE2L2 (0.39) TRIM24TRIM33KDM4EKMT2ANPSR1
SCHEMBL2674974 0.78 KDM4E (0.36) TRIM24TRIM33KDM4ENPSR1L3MBTL1
SCHEMBL28191855 0.78 KDM4E (0.47) KDM4EKMT2ANPSR1L3MBTL1MEN1
SCHEMBL2561503 0.77 L3MBTL1 (0.57) TRIM24TRIM33KDM4EKMT2ANPSR1
SCHEMBL14097048 0.77 PLK1 (0.46) TRIM24TRIM33KDM4EKMT2ANPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2225238-B1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZOÝ1,2- ¨IMIDAZOLE-3- CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INT (DE) 2014-09-03 EP disclosed
US-8552205-B2 Derivatives of 6,7-dihydro-5H-imidazo[1,2-alpha]imidazole-3-carboxylic acid amides BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2013-10-08 US disclosed
US-20110224188-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-alpha]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2011-09-15 US disclosed
EP-2225238-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZOÝ1,2- ¨IMIDAZOLE-3- CARBOXYLIC ACID AMIDES Boehringer Ingelheim International GmbH (DE) 2010-09-08 EP disclosed
WO-2009070485-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-α]IMIDAZOLE-3- CARBOXYLIC ACID AMIDES BOEHRINGER INGELHEIM INTERNATIONAL GMBH (DE) 2009-06-04 WO disclosed
US-5262387-A Pyridine derivatives and their use for controlling undesirable plant growth BASF AKTIENGESELLSCHAFT (DE) 1993-11-16 US disclosed
US-5262384-A Herbicides BASF AKTIENGESELLSCHAFT (DE) 1993-11-16 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110224188-A1 DERIVATIVES OF 6,7-DIHYDRO-5H-IMIDAZO[1,2-alpha]IMIDAZOLE-3-CARBOXYLIC ACID AMIDES HPGDS, COL14A1, ARG1 TRIM24 493/4885TRIM33 1507/4885KDM4E 1701/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.