SCHEMBL2394586

SCHEMBL2394586

ON=C(COc1cccnc1)c1ccccc1

nearest known ligand 0.53

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
MAPT P10636 1/20 0.51
NOTUM Q6P988 1/20 0.47
CHRNB2 P17787 4/20 0.46
CHRNA4 P43681 4/20 0.46
NAMPT P43490 1/20 0.45
GALR3 O60755 1/20 0.44
RAB9A P51151 1/20 0.44
TDP1 Q9NUW8 1/20 0.44
HTT P42858 1/20 0.41
PLOD2 O00469 1/20 0.41
GAA P10253 1/20 0.41
CYP11B1 P15538 1/20 0.41
CYP11B2 P19099 1/20 0.41
DRD4 P21917 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2394579 1.00 MAPT (0.51) MAPTNOTUMCHRNB2CHRNA4NAMPT
SCHEMBL31351884 0.85 ALOX15 (0.50) MAPTGAADRD4
SCHEMBL2394339 0.82 MAPT (0.47) MAPTNOTUMCHRNB2CHRNA4NAMPT
SCHEMBL2394334 0.82 MAPT (0.47) MAPTNOTUMCHRNB2CHRNA4NAMPT
SCHEMBL2394585 0.79 PLOD2 (0.58) MAPTNOTUMNAMPTGALR3RAB9A
SCHEMBL2009003 0.75 ALOX15 (0.62) MAPTNOTUMCHRNB2CHRNA4NAMPT
SCHEMBL9323799 0.74 NAPRT (0.54) RAB9ATDP1HTTPLOD2GAA
SCHEMBL9323795 0.74 NAPRT (0.54) RAB9ATDP1HTTPLOD2GAA
SCHEMBL20491186 0.74 GAA (0.50) MAPTGAADRD4
SCHEMBL2396340 0.74 SLC6A4 (0.51) MAPTGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed