SCHEMBL23958208

SCHEMBL23958208

Cc1ccccc1-n1c(Nc2cccnc2)nc2ccc(F)cc2c1=O

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TDO2 P48775 2/20 0.48
IDO2 Q6ZQW0 2/20 0.48
PDE7A Q13946 1/20 0.46
PDE4D Q08499 1/20 0.44
TP53 P04637 1/20 0.44
PI4KA P42356 1/20 0.43
PIK3CG P48736 1/20 0.43
ALDH1A1 P00352 2/20 0.43
LMNA P02545 2/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
IDO1 P14902 1/20 0.42
KDM4E B2RXH2 1/20 0.42
MAPT P10636 1/20 0.42
G6PD P11413 1/20 0.42
PKM P14618 1/20 0.42
MPI P34949 1/20 0.42
HTT P42858 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.42
HDAC8 Q9BY41 1/20 0.42
APOBEC3G Q9HC16 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30103275 1.00 TDO2 (0.48) TDO2IDO2PDE7APDE4DTP53
SCHEMBL23958346 0.92 PDE7A (0.46) TDO2IDO2PDE7ATP53ALDH1A1
SCHEMBL30103212 0.91 TDO2 (0.48) TDO2IDO2L3MBTL1IDO1
SCHEMBL23958205 0.91 TDO2 (0.48) TDO2IDO2L3MBTL1IDO1
SCHEMBL29423292 0.89 TDO2 (0.49) TDO2IDO2PDE4DTP53PI4KA
SCHEMBL24110983 0.89 TDO2 (0.49) TDO2IDO2PDE4DTP53PI4KA
SCHEMBL30103195 0.88 HTR7 (0.46) TDO2IDO2TP53LMNAL3MBTL1
SCHEMBL23958283 0.88 HTR7 (0.46) TDO2IDO2TP53LMNAL3MBTL1
SCHEMBL23958262 0.88
SCHEMBL30103230 0.88

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115427399-A 2-heteroarylaminoquinazolinone derivatives 住友制药株式会社 2022-12-02 CN disclosed
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-16 US disclosed
WO-2021215537-A1 2-HETEROARYLAMINOQUINAZOLINONE DERIVATIVE 大日本住友製薬株式会社 (JP) 2021-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE CRKL, CLIC4, CLIC1 TDO2 1621/4885IDO2 443/4885PDE7A 3371/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.