SCHEMBL23958283

SCHEMBL23958283

COc1ccccc1-n1c(Nc2cccnc2)nc2ccc(F)cc2c1=O

nearest known ligand 0.54

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR7 P34969 3/20 0.46
ALPL P05186 1/20 0.44
TDO2 P48775 1/20 0.44
IDO2 Q6ZQW0 1/20 0.44
TP53 P04637 2/20 0.44
LMNA P02545 1/20 0.44
L3MBTL1 Q9Y468 1/20 0.43
HTR1A P08908 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2C P28335 1/20 0.43
POLB P06746 1/20 0.42
MAPT P10636 1/20 0.42
HPD P32754 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30103195 1.00 HTR7 (0.46) HTR7ALPLTDO2IDO2TP53
SCHEMBL23958205 0.89 TDO2 (0.48) TDO2IDO2L3MBTL1
SCHEMBL30103212 0.89 TDO2 (0.48) TDO2IDO2L3MBTL1
SCHEMBL30103275 0.88 TDO2 (0.48) TDO2IDO2TP53LMNAL3MBTL1
SCHEMBL23958208 0.88 TDO2 (0.48) TDO2IDO2TP53LMNAL3MBTL1
SCHEMBL23958262 0.86
SCHEMBL30103230 0.86
SCHEMBL23958265 0.86 PIK3CD (0.46) TDO2IDO2POLB
SCHEMBL29738614 0.86 PIK3CD (0.46) TDO2IDO2POLB
SCHEMBL24110985 0.85 G6PD (0.50) HTR7LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115427399-A 2-heteroarylaminoquinazolinone derivatives 住友制药株式会社 2022-12-02 CN disclosed
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-16 US disclosed
WO-2021215537-A1 2-HETEROARYLAMINOQUINAZOLINONE DERIVATIVE 大日本住友製薬株式会社 (JP) 2021-10-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE CRKL, CLIC4, CLIC1 HTR7 1211/4885ALPL 4100/4885TDO2 1621/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.