SCHEMBL23958797

SCHEMBL23958797

COc1cc(C(=O)NCC(c2cc(C(C)(C)O)c(F)c(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C(F)(F)F)cnc12

nearest known ligand 0.53

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.36
LMNA P02545 1/20 0.33
TP53 P04637 1/20 0.33
PDE4B Q07343 2/20 0.33
P2RX7 Q99572 3/20 0.33
HCRTR1 O43613 3/20 0.32
HCRTR2 O43614 1/20 0.32
ALDH1A1 P00352 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
ACSS2 Q9NR19 1/20 0.32
ROCK2 O75116 3/20 0.32
ROCK1 Q13464 3/20 0.32
GABRA5 P31644 1/20 0.32
ALOX5 P09917 1/20 0.31
EPHX2 P34913 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958810 0.94 CFTR (0.34) CFTRLMNATP53PDE4BP2RX7
SCHEMBL23958776 0.90 LMNA (0.36) CFTRLMNATP53PDE4BP2RX7
SCHEMBL23958652 0.90 LMNA (0.33) CFTRLMNATP53ALDH1A1SMN1; SMN2
SCHEMBL23958859 0.86 CFTR (0.34) CFTRLMNATP53ALDH1A1SMN1; SMN2
SCHEMBL25698171 0.85 PDE4B (0.31) PDE4BACSS2
SCHEMBL23958874 0.85 CTSA (0.35) PDE4BACSS2ROCK2ROCK1GABRA5
SCHEMBL23958656 0.84 SSTR5 (0.34) EPHX2
SCHEMBL25698133 0.84 PDE4B (0.35) PDE4BP2RX7HCRTR1HCRTR2ACSS2
SCHEMBL26766103 0.83 IRAK4 (0.39) CFTRLMNATP53
SCHEMBL25687503 0.82 CFTR (0.38) CFTRPDE4BHCRTR1HCRTR2ROCK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed