SCHEMBL23958776

SCHEMBL23958776

COc1cc(C(=O)NCC(c2cc(C(C)(C)O)c(F)c(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C(F)F)cnc12

nearest known ligand 0.51

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.36
TP53 P04637 1/20 0.36
ALDH1A1 P00352 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
P2RX7 Q99572 8/20 0.34
IRAK4 Q9NWZ3 1/20 0.34
CFTR P13569 3/20 0.33
KCNH2 Q12809 2/20 0.32
FFAR1 O14842 1/20 0.32
PDE4B Q07343 1/20 0.31
ROCK2 O75116 1/20 0.31
ROCK1 Q13464 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958652 0.90 LMNA (0.33) LMNATP53ALDH1A1SMN1; SMN2IRAK4
SCHEMBL23958797 0.90 CFTR (0.36) LMNATP53ALDH1A1SMN1; SMN2P2RX7
SCHEMBL23958859 0.86 CFTR (0.34) LMNATP53ALDH1A1SMN1; SMN2CFTR
SCHEMBL25698171 0.85 PDE4B (0.31) IRAK4PDE4B
SCHEMBL23958874 0.85 CTSA (0.35) FFAR1PDE4BROCK2ROCK1
SCHEMBL23958810 0.84 CFTR (0.34) LMNATP53SMN1; SMN2P2RX7CFTR
SCHEMBL26766103 0.83 IRAK4 (0.39) LMNATP53IRAK4CFTRKCNH2
SCHEMBL30007232 0.83 CFTR (0.34) LMNATP53ALDH1A1SMN1; SMN2P2RX7
SCHEMBL25687300 0.83 CFTR (0.34) LMNATP53ALDH1A1SMN1; SMN2P2RX7
SCHEMBL25687497 0.81 CFTR (0.38) CFTR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed