SCHEMBL23958810

SCHEMBL23958810

COc1cc(C(=O)NCC(c2cc(C(C)(C)O)c(Cl)c(-c3ccc(F)cc3)n2)C2CC2)cc2cc(C(F)(F)F)cnc12

nearest known ligand 0.46

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.34
P2RX7 Q99572 9/20 0.34
LMNA P02545 1/20 0.32
TP53 P04637 1/20 0.32
DDR1 Q08345 1/20 0.32
PDE4B Q07343 2/20 0.32
HCRTR1 O43613 1/20 0.31
HCRTR2 O43614 1/20 0.31
MAPT P10636 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
CCR5 P51681 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958797 0.94 CFTR (0.36) CFTRP2RX7LMNATP53PDE4B
SCHEMBL23958990 0.87 CFTR (0.33) CFTRP2RX7LMNATP53DDR1
SCHEMBL23958786 0.85 IRAK4 (0.32) CFTRP2RX7LMNAMAPT
SCHEMBL23958776 0.84 LMNA (0.36) CFTRP2RX7LMNATP53PDE4B
SCHEMBL23958652 0.84 LMNA (0.33) CFTRLMNATP53MAPTSMN1; SMN2
SCHEMBL25698156 0.84 PDE4B (0.34) P2RX7PDE4B
SCHEMBL25687507 0.83 CFTR (0.36) CFTRP2RX7PDE4BHCRTR1HCRTR2
SCHEMBL28909199 0.83 CFTR (0.36) CFTRP2RX7PDE4BHCRTR1HCRTR2
SCHEMBL23958726 0.81 CFTR (0.35) CFTRLMNATP53MAPTSMN1; SMN2
SCHEMBL25687501 0.81 CFTR (0.39) CFTRDDR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed