SCHEMBL23958812

SCHEMBL23958812

COc1cc(C(=O)NCC(O)c2cc(C(C)(C)O)c(F)c(-c3ccc(F)cc3)n2)cc(/C=C(/C)N)c1N

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.38
MAPT P10636 2/20 0.34
ALDH1A1 P00352 3/20 0.34
POLB P06746 2/20 0.34
KDM4E B2RXH2 2/20 0.34
RECQL P46063 1/20 0.34
KMT2A Q03164 1/20 0.33
CNR2 P34972 2/20 0.32
SCN9A Q15858 2/20 0.32
BTK Q06187 1/20 0.32
ROCK2 O75116 2/20 0.32
ROCK1 Q13464 2/20 0.32
ACSS2 Q9NR19 1/20 0.32
GAA P10253 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958802 0.88 CFTR (0.34) CFTRMAPTALDH1A1POLBKDM4E
SCHEMBL23958782 0.84 CFTR (0.35) CFTRMAPTALDH1A1POLBKDM4E
SCHEMBL23958976 0.84 KDM4E (0.31) CFTRMAPTALDH1A1POLBKDM4E
SCHEMBL23958775 0.84 ADRA1D (0.36) CFTRMAPTALDH1A1POLBKDM4E
SCHEMBL23958792 0.80 CFTR (0.33) CFTRMAPTALDH1A1POLBKDM4E
SCHEMBL23958753 0.78 CFTR (0.32) CFTR
SCHEMBL23958813 0.77 CFTR (0.32) CFTR
SCHEMBL23958894 0.77 CFTR (0.34) CFTRMAPTALDH1A1POLBKDM4E
SCHEMBL23958834 0.76 CFTR (0.35) CFTR
SCHEMBL23904891 0.75 PTGS1 (0.33) CFTRMAPTALDH1A1POLBKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed