SCHEMBL23958775

SCHEMBL23958775

COc1cc(C(=O)NCC(c2cc(C(C)(C)O)c(F)c(-c3ccc(C(F)(F)F)cc3)n2)C2CC2)cc(/C=C(/C)N)c1N

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 2/20 0.36
ADRA1A P35348 2/20 0.36
ADRA1B P35368 2/20 0.36
MAPT P10636 3/20 0.34
CFTR P13569 3/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
ROCK2 O75116 1/20 0.32
ROCK1 Q13464 1/20 0.32
PDE2A O00408 1/20 0.31
BTK Q06187 1/20 0.31
KDM4E B2RXH2 1/20 0.31
ALDH1A1 P00352 1/20 0.31
POLB P06746 1/20 0.31
RECQL P46063 1/20 0.31
MTTP P55157 1/20 0.31
EPHX2 P34913 1/20 0.30
PPARG P37231 1/20 0.30
PPARD Q03181 1/20 0.30
PPARA Q07869 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958976 0.92 KDM4E (0.31) MAPTCFTRKDM4EALDH1A1POLB
SCHEMBL23958782 0.88 CFTR (0.35) MAPTCFTRSMN1; SMN2KDM4EALDH1A1
SCHEMBL23958802 0.86 CFTR (0.34) MAPTCFTRROCK2ROCK1KDM4E
SCHEMBL23958812 0.84 CFTR (0.38) MAPTCFTRROCK2ROCK1BTK
SCHEMBL23905980 0.83 ADRA1D (0.33) ADRA1DADRA1AADRA1BMAPTSMN1; SMN2
SCHEMBL23958753 0.82 CFTR (0.32) CFTR
SCHEMBL23958792 0.81 CFTR (0.33) MAPTCFTRSMN1; SMN2ROCK2ROCK1
SCHEMBL23958894 0.81 CFTR (0.34) MAPTCFTRSMN1; SMN2KDM4EALDH1A1
SCHEMBL23958797 0.80 CFTR (0.36) CFTRSMN1; SMN2ROCK2ROCK1ALDH1A1
SCHEMBL23958739 0.76 TRPV3 (0.34) CFTRPDE2AMDM2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed