SCHEMBL23958894

SCHEMBL23958894

COc1cc(C(=O)NCC(c2cc(C(C)(C)O)c(Cl)c(-c3ccc(F)cc3)n2)C2CC2)cc(/C=C(\N)C(F)F)c1N

nearest known ligand 0.37

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
CFTR P13569 3/20 0.34
MAPT P10636 3/20 0.31
ALDH1A1 P00352 3/20 0.31
LMNA P02545 1/20 0.31
TP53 P04637 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
DDR1 Q08345 1/20 0.31
KDM4E B2RXH2 2/20 0.30
POLB P06746 2/20 0.30
RECQL P46063 1/20 0.30
TLR9 Q9NR96 1/20 0.30
TLR8 Q9NR97 1/20 0.30
TLR7 Q9NYK1 1/20 0.30
P2RX7 Q99572 1/20 0.30
MEN1 O00255 1/20 0.30
GAA P10253 1/20 0.30
HPGD P15428 1/20 0.30
KMT2A Q03164 1/20 0.30
HTR4 Q13639 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23958782 0.93 CFTR (0.35) CFTRMAPTALDH1A1LMNATP53
SCHEMBL23958753 0.89 CFTR (0.32) CFTR
SCHEMBL23958775 0.81 ADRA1D (0.36) CFTRMAPTALDH1A1SMN1; SMN2KDM4E
SCHEMBL23958976 0.81 KDM4E (0.31) CFTRMAPTALDH1A1KDM4EPOLB
SCHEMBL23958990 0.81 CFTR (0.33) CFTRMAPTALDH1A1LMNATP53
SCHEMBL23958810 0.80 CFTR (0.34) CFTRMAPTLMNATP53SMN1; SMN2
SCHEMBL23958802 0.80 CFTR (0.34) CFTRMAPTALDH1A1KDM4EPOLB
SCHEMBL23958779 0.79 MAPT (0.33) MAPTALDH1A1LMNATP53SMN1; SMN2
SCHEMBL23958792 0.78 CFTR (0.33) CFTRMAPTALDH1A1LMNATP53
SCHEMBL23958812 0.77 CFTR (0.38) CFTRMAPTALDH1A1KDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021214136-A1 RSV INHIBITING 3-SUBSTITUTED QUINOLINE AND CINNOLINE DERIVATIVES Janssen Sciences Ireland Unlimited Company (IE) 2021-10-28 WO disclosed