SCHEMBL23964667

SCHEMBL23964667

CC(Cc1cc(I)c(O)c(I)c1)C(=O)O

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SIRT5 Q9NXA8 1/20 0.55
CYP2C9 P11712 2/20 0.54
CYP2C19 P33261 1/20 0.54
HIF1A Q16665 1/20 0.54
THRB P10828 6/20 0.51
MEN1 O00255 4/20 0.51
KMT2A Q03164 4/20 0.51
PPARG P37231 4/20 0.51
THRA P10827 4/20 0.51
LMNA P02545 2/20 0.51
TTR P02766 2/20 0.51
ADORA3 P0DMS8 2/20 0.51
PDE4D Q08499 2/20 0.51
HSD17B10 Q99714 2/20 0.51
NR1I2 O75469 2/20 0.51
RXRA P19793 2/20 0.51
NR3C1 P04150 1/20 0.51
CYP1A2 P05177 1/20 0.51
HTR1A P08908 1/20 0.51
TBXA2R P21731 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3217395 0.86 THRB (0.73) CYP2C9HIF1ATHRBMEN1KMT2A
SCHEMBL12200634 0.85 LMNA (0.48) SIRT5CYP2C9CYP2C19HIF1ATHRB
SCHEMBL12200628 0.82 FOLH1 (0.59) CYP2C9CYP2C19HIF1ATHRBMEN1
SCHEMBL11225864 0.81 SIRT5 (0.55) SIRT5CYP2C9CYP2C19HIF1ATHRB
SCHEMBL9972708 0.81 HMGB1 (0.46) SIRT5CYP2C9CYP2C19HIF1ATHRB
SCHEMBL5858308 0.79 PTPN1 (0.44) SIRT5CYP2C9CYP2C19HIF1ATHRB
SCHEMBL14032679 0.79 FFAR4 (0.41) SIRT5CYP2C9CYP2C19HIF1APTGS2
Diotyrosine SCHEMBL147578 0.79 SIRT5 (0.82) SIRT5CYP2C9THRBMEN1KMT2A
Diotyrosine SCHEMBL838215 0.79 SIRT5 (0.82) SIRT5CYP2C9THRBMEN1KMT2A
Diotyrosine SCHEMBL147579 0.79 SIRT5 (0.82) SIRT5CYP2C9THRBMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021216529-A1 β-ARRESTIN EFFECTORS AND COMPOSITIONS AND METHODS OF USE THEREOF TREVENA, INC. (US) 2021-10-28 WO disclosed