SCHEMBL2396587

SCHEMBL2396587

COc1ccc(SC[C@@H](N)c2ccccc2)cc1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN4A P35499 5/20 0.51
CYP1A2 P05177 1/20 0.47
CYP2D6 P10635 1/20 0.47
CYP2C19 P33261 1/20 0.47
MAOA P21397 1/20 0.47
MAOB P27338 1/20 0.47
NPC1 O15118 1/20 0.45
KIF11 P52732 4/20 0.43
TACR1 P25103 1/20 0.43
EPHX1 P07099 1/20 0.43
ALDH1A1 P00352 1/20 0.41
ACP3 P15309 1/20 0.41
PBRM1 Q86U86 1/20 0.41
CA4 P22748 1/20 0.41
LTA4H P09960 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9299256 0.82 MAOA (0.61) SCN4AMAOAMAOBALDH1A1
SCHEMBL1496515 0.81 SMN1; SMN2 (0.46) NPC1EPHX1ALDH1A1ACP3CA4
SCHEMBL28915703 0.78 L3MBTL1 (0.46) NPC1KIF11EPHX1ALDH1A1ACP3
SCHEMBL28915705 0.78 L3MBTL1 (0.46) NPC1KIF11EPHX1ALDH1A1ACP3
SCHEMBL15326789 0.75 SCN4A (0.76) SCN4ACYP1A2CYP2D6CYP2C19TACR1
SCHEMBL5680007 0.75 CYP1A2 (0.83) CYP1A2CYP2D6CYP2C19TACR1EPHX1
SCHEMBL1255723 0.74 KIF11 (0.67) CYP1A2CYP2D6CYP2C19KIF11
SCHEMBL28825153 0.74 LMNA (0.55) NPC1EPHX1ALDH1A1
SCHEMBL24019096 0.73 NPC1 (0.51) CYP1A2CYP2D6CYP2C19MAOAMAOB
SCHEMBL9768891 0.73 CA4 (0.44) MAOAMAOBNPC1ALDH1A1CA4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed
US-8012901-B1 Method of synthesizing enantiopure mexiletine analogues and novel β-thiophenoxy and pyridyl ethers NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2011-09-06 US disclosed