SCHEMBL23969189

SCHEMBL23969189

C=C(CCc1ccc(C)cc1C(=O)CC)NCCNC

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
ALDH1A1 P00352 3/20 0.33
HPGD P15428 2/20 0.33
TSHR P16473 1/20 0.33
HSD17B10 Q99714 1/20 0.33
SMN1; SMN2 Q16637 3/20 0.33
HTT P42858 2/20 0.33
MMP2 P08253 1/20 0.32
MMP9 P14780 1/20 0.32
ADAM17 P78536 1/20 0.32
LMNA P02545 1/20 0.31
KDM4E B2RXH2 1/20 0.31
CYP3A4 P08684 1/20 0.31
NPC1 O15118 1/20 0.30
RAB9A P51151 1/20 0.30
MTNR1A P48039 1/20 0.30
MTNR1B P49286 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL22175873 0.88
SCHEMBL23969316 0.87 MTNR1A (0.37) LMNAKDM4ECYP3A4MTNR1A
SCHEMBL22175941 0.83 ALDH1A1 (0.39) MEN1KMT2AALDH1A1HPGDTSHR
SCHEMBL22175868 0.77 GABRG2 (0.31) ALDH1A1HPGDTSHRHSD17B10
SCHEMBL22175888 0.77 ALDH1A1 (0.41) ALDH1A1HPGDHTTLMNAKDM4E
SCHEMBL23969190 0.75
SCHEMBL23969380 0.75
SCHEMBL22175855 0.75 HTT (0.37) HPGDTSHRSMN1; SMN2HTTLMNA
SCHEMBL23969192 0.74 MTNR1A (0.34) ALDH1A1HPGDTSHRHSD17B10SMN1; SMN2
SCHEMBL22175867 0.73 GABRG2 (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3903788-A1 PYRAZOLO[1,5-A]PYRIMIDINE MACROCYCLIC COMPOUND Taisho Pharmaceutical Co., Ltd. (JP) 2021-11-03 EP disclosed