SCHEMBL23972809

SCHEMBL23972809

Cc1ccc(C2(C(=N)N)CC2)cc1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 4/20 0.39
MAOA P21397 2/20 0.39
IDO1 P14902 2/20 0.38
CYP3A4 P08684 1/20 0.38
CYP2D6 P10635 1/20 0.38
CYP2C9 P11712 1/20 0.38
HSD11B1 P28845 1/20 0.38
OPRM1 P35372 2/20 0.37
WDR5 P61964 1/20 0.37
OPRK1 P41145 1/20 0.35
OPRL1 P41146 1/20 0.35
HTR3E A5X5Y0 1/20 0.34
SLC22A2 O15244 1/20 0.34
SLC22A1 O15245 1/20 0.34
SLC22A3 O75751 1/20 0.34
HTR3B O95264 1/20 0.34
PLAU P00749 1/20 0.34
HTR3A P46098 1/20 0.34
HTR3D Q70Z44 1/20 0.34
HTR3C Q8WXA8 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL171875 0.79 LMNA (0.47) MAOBMAOACYP3A4CYP2D6CYP2C9
SCHEMBL1622891 0.78 AKR1C1 (0.47) MAOBMAOAHSD11B1
Hydrochloric Acid SCHEMBL435506 0.78 OPRM1 (0.46) MAOBMAOACYP3A4CYP2D6CYP2C9
Hydrochloric Acid SCHEMBL28933139 0.77 AKR1C1 (0.45) MAOBMAOAHSD11B1
SCHEMBL23972282 0.76 ADRA2A (0.40) IDO1SPHK2SPHK1
SCHEMBL23972810 0.75 MAOA (0.46) MAOBMAOAIDO1OPRM1OPRL1
Acetic Acid SCHEMBL17102034 0.74 NQO2 (0.43) CYP3A4CYP2C9HSD11B1OPRM1MAPT
SCHEMBL2701195 0.73 MAPT (0.46) MAPTTDP1
SCHEMBL5379326 0.72 HSD11B1 (0.45) CYP3A4CYP2D6CYP2C9HSD11B1OPRM1
SCHEMBL351393 0.72 AKR1C1 (0.55) CYP3A4CYP2D6CYP2C9HSD11B1OPRM1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2021221169-A1 PYRIMIDIN-4(3H)-ONE DERIVATIVES AS TRPV4 ANTAGONISTS RAQUALIA PHARMA INC. (JP) 2021-11-04 WO disclosed