SCHEMBL24019233

SCHEMBL24019233

COC(=O)c1cc(I)c2nc(C)cnc2c1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATM Q13315 1/20 0.43
KDM4E B2RXH2 5/20 0.41
ALDH1A1 P00352 4/20 0.41
CSNK2A1 P68400 1/20 0.38
HPGD P15428 3/20 0.38
MEN1 O00255 2/20 0.38
KMT2A Q03164 2/20 0.38
ALOX15 P16050 1/20 0.38
HTT P42858 1/20 0.38
CA12 O43570 1/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
CA7 P43166 1/20 0.38
CA9 Q16790 1/20 0.38
CA14 Q9ULX7 1/20 0.38
RXFP1 Q9HBX9 1/20 0.38
PSMD14 O00487 1/20 0.37
L3MBTL1 Q9Y468 2/20 0.37
LMNA P02545 1/20 0.37
POLB P06746 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23905568 0.83 KDM4E (0.45) ATMKDM4EALDH1A1CSNK2A1HPGD
SCHEMBL17442622 0.75 ATM (0.51) ATMKDM4EALDH1A1HPGDMEN1
SCHEMBL17442654 0.71 PSMD14 (0.43) ATMKDM4EALDH1A1CSNK2A1HPGD
SCHEMBL29940501 0.70 KDM4E (0.41) ATMKDM4EALDH1A1HPGDALOX15
SCHEMBL29278006 0.70 KDM4E (0.41) ATMKDM4EALDH1A1HPGDALOX15
SCHEMBL18739565 0.70
SCHEMBL24019244 0.70 HSD17B10 (0.34)
SCHEMBL23905769 0.70 CA12 (0.47) KMT2AALOX15HTTCA12CA1
SCHEMBL17442548 0.70 ALOX15 (0.58) KDM4EALDH1A1HPGDMEN1KMT2A
SCHEMBL24019234 0.69 OGA (0.30)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3359533-B1 QUINOXALINE AND PYRIDOPYRAZINE DERIVATIVES AS PI3KBETA INHIBITORS JANSSEN PHARMACEUTICA NV (BE) 2021-11-17 EP disclosed