SCHEMBL2403262

SCHEMBL2403262

COc1ccc2[nH]c(C(C)=O)c(CCN)c2c1

nearest known ligand 0.65

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 1/20 0.65
HTR6 P50406 1/20 0.65
ALDH1A1 P00352 4/20 0.62
KDM4E B2RXH2 3/20 0.62
HPGD P15428 3/20 0.62
HSD17B10 Q99714 2/20 0.62
POLB P06746 1/20 0.60
MDM2 Q00987 1/20 0.60
NQO2 P16083 3/20 0.56
MTNR1A P48039 12/20 0.55
MTNR1B P49286 12/20 0.55
AKR1C2 P52895 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP3A4 P08684 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
CYP2C19 P33261 1/20 0.52
NPC1 O15118 1/20 0.51
MAPT P10636 1/20 0.51

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28793909 0.88 HTR6 (0.50) HTR1DHTR6ALDH1A1KDM4EHPGD
SCHEMBL16716149 0.86 HTR1D (0.61) HTR1DHTR6ALDH1A1KDM4EHPGD
Hydrochloric Acid SCHEMBL16711692 0.85 HTR1D (0.60) HTR1DHTR6ALDH1A1KDM4EHPGD
SCHEMBL27566660 0.85 NQO2 (0.72) HTR1DHTR6ALDH1A1KDM4EHPGD
SCHEMBL6948872 0.84 KDM4E (0.58) HTR1DHTR6ALDH1A1KDM4EHPGD
SCHEMBL3221458 0.84 KDM4E (0.84) ALDH1A1KDM4EHPGDHSD17B10POLB
SCHEMBL1345727 0.82 KDM4E (0.73) HTR1DHTR6ALDH1A1KDM4EHPGD
SCHEMBL6950433 0.82 ALDH1A1 (0.70) ALDH1A1KDM4EHPGDHSD17B10POLB
Hydrochloric Acid SCHEMBL1343869 0.81 ALDH1A1 (0.72) HTR1DHTR6ALDH1A1KDM4EHPGD
SCHEMBL4244966 0.79 HTR1D (1.00) HTR1DHTR6ALDH1A1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011112167-A1 COMPOSITIONS AND METHODS FOR DIABETES TREATMENT RESET THERAPEUTICS, INC. (US) 2011-09-15 WO disclosed