SCHEMBL24038698

SCHEMBL24038698

CCOC(=O)C1c2ccc(S(=O)(=O)CC3CC3)cc2CCN1C(=O)OC(C)(C)C

nearest known ligand 0.49

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
RORC P51449 4/20 0.49
GPR119 Q8TDV5 3/20 0.43
GHSR Q92847 13/20 0.42
CYP2D6 P10635 1/20 0.41
KCNH2 Q12809 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30920109 0.92 GHSR (0.45) GPR119GHSR
SCHEMBL24031466 0.92 GHSR (0.45) GPR119GHSR
SCHEMBL24038710 0.89 GHSR (0.46) RORCGPR119GHSRCYP2D6KCNH2
SCHEMBL24031031 0.88 GPR119 (0.49) RORCGPR119GHSR
SCHEMBL24038697 0.87 GHSR (0.46) GPR119GHSR
SCHEMBL25895663 0.82 GHSR (0.46) GHSR
SCHEMBL17391030 0.82 GHSR (0.54) GHSR
SCHEMBL17391103 0.82 GHSR (0.57) GHSR
SCHEMBL2081445 0.81 ESR2 (0.49) GHSR
SCHEMBL24031477 0.81 GHSR (0.49) GPR119GHSR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-118580188-A Can be used as ROR gamma regulator aniline compound (B) 励缔(杭州)医药科技有限公司 2024-09-03 CN disclosed
CN-113773251-B Anilines useful as rory modulators 励缔(杭州)医药科技有限公司 2024-06-11 CN disclosed
US-20230192620-A1 ANILINE COMPOUND USED AS RORy REGULATOR SHANGHAI LITEDD CO., LTD. (CN) 2023-06-22 US disclosed
US-20230192620-A1 ANILINE COMPOUND USED AS RORy REGULATOR SHANGHAI LITEDD CO., LTD. (CN) 2023-06-22 US disclosed
CN-113773251-A Anilines useful as ROR gamma modulators 上海辉启生物医药科技有限公司 2021-12-10 CN disclosed
WO-2021228217-A1 ANILINE COMPOUND USED AS RORγ REGULATOR 上海辉启生物医药科技有限公司 2021-11-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20230192620-A1 ANILINE COMPOUND USED AS RORy REGULATOR RORB, RORA, RORC RORC 3/4885GPR119 240/4885GHSR 691/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.