SCHEMBL2407587

SCHEMBL2407587

CC(C)(C)CN(Cc1cn(S(=O)(=O)c2ccccc2)c(-c2cccnc2C(F)(F)F)c1F)C(=O)O

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.34
PTGDR2 Q9Y5Y4 5/20 0.34
HTR6 P50406 4/20 0.34
CHRM5 P08912 1/20 0.32
NR1I2 O75469 3/20 0.32
CCNE1 P24864 1/20 0.31
CDK2 P24941 1/20 0.31
HSD11B1 P28845 1/20 0.31
MET P08581 1/20 0.31
CYP2C19 P33261 1/20 0.31
RORA P35398 1/20 0.31
RORC P51449 1/20 0.31
RORB Q92753 1/20 0.31
NR1H4 Q96RI1 1/20 0.31
KDM4E B2RXH2 1/20 0.30
ALDH1A1 P00352 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2408646 0.93 RORC (0.33) DHODHPTGDR2HTR6CHRM5RORC
SCHEMBL2412422 0.89 PTGDR2 (0.34) DHODHPTGDR2HTR6METCYP2C19
SCHEMBL4999141 0.88 HTR6 (0.37) DHODHPTGDR2HTR6CCNE1CDK2
SCHEMBL2410603 0.86 HTR6 (0.33) PTGDR2HTR6CHRM5METCYP2C19
SCHEMBL2409445 0.85 ESR1 (0.39) PTGDR2HTR6
SCHEMBL2411045 0.84 PTGER2 (0.33) PTGDR2HTR6RORCKDM4E
SCHEMBL4420273 0.84 HTR6 (0.36) PTGDR2HTR6
SCHEMBL2413762 0.83 SLC6A9 (0.35) PTGDR2HTR6CHRM5RORC
SCHEMBL2407589 0.83 MET (0.39) PTGDR2HTR6CHRM5MET
SCHEMBL2407583 0.83 SOS1 (0.36) DHODHPTGDR2HTR6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed