SCHEMBL2409441

SCHEMBL2409441

CN(Cc1cn(S(=O)(=O)c2ccc(O)cc2)c(-c2cccnc2F)c1F)C(=O)OC(C)(C)C

nearest known ligand 0.35

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTR2C P28335 6/20 0.35
SLC6A4 P31645 6/20 0.35
KAT6A Q92794 2/20 0.34
KAT5 Q92993 2/20 0.34
HTR2A P28223 1/20 0.33
KAT8 Q9H7Z6 2/20 0.33
MMP2 P08253 2/20 0.32
MMP9 P14780 2/20 0.32
MMP8 P22894 2/20 0.32
MMP13 P45452 2/20 0.32
SSTR4 P31391 1/20 0.31
HTR6 P50406 1/20 0.31
PDK2 Q15119 1/20 0.30
F2 P00734 1/20 0.30
ESR1 P03372 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL4424124 0.94 KAT6A (0.34) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL1833792 0.90 KAT6A (0.32) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL2411207 0.90 HTR6 (0.39) HTR2CSLC6A4KAT6AKAT5MMP2
SCHEMBL2411042 0.89 HTR6 (0.33) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL4420269 0.88 HTR6 (0.37) HTR2CSLC6A4HTR2AKAT8HTR6
SCHEMBL1834426 0.88 HTR2C (0.33) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL4570001 0.88 OXTR (0.34) HTR2CSLC6A4KAT6AKAT5MMP2
SCHEMBL2412512 0.87 HTR2C (0.31) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL2408895 0.87 SSTR4 (0.32) HTR2CSLC6A4KAT6AKAT5HTR2A
SCHEMBL2407588 0.87 MET (0.38) HTR2CSLC6A4KAT6AKAT5HTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2364979-A1 Pyrrole compounds Takeda Pharmaceutical Company Limited (JP) 2011-09-14 EP disclosed
EP-2114917-A2 PYRROLE COMPOUNDS Takeda Pharmaceutical Company Limited (JP) 2009-11-11 EP disclosed
WO-2008108380-A2 PYRROLE COMPOUNDS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2008-09-12 WO disclosed