SCHEMBL24080922

SCHEMBL24080922

CN1C(=O)Cc2c(S)cccc21

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRPF1 P55201 1/20 0.40
CCNB2 O95067 1/20 0.38
CDK1 P06493 1/20 0.38
CCNB1 P14635 1/20 0.38
GSK3B P49841 1/20 0.38
CCNB3 Q8WWL7 1/20 0.38
KMT2A Q03164 4/20 0.36
MEN1 O00255 3/20 0.36
OPRL1 P41146 2/20 0.35
OPRK1 P41145 1/20 0.35
PDE4D Q08499 1/20 0.35
GABRA1 P14867 1/20 0.34
GABRG2 P18507 1/20 0.34
GABRB3 P28472 1/20 0.34
GABRA5 P31644 1/20 0.34
CCKBR P32239 1/20 0.34
GABRA3 P34903 1/20 0.34
GABRA2 P47869 1/20 0.34
GABRB2 P47870 1/20 0.34
MAPT P10636 2/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL256751 0.79 KMT2A (0.46) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL19704723 0.79 SMN1; SMN2 (0.42) KMT2AMEN1MAPT
SCHEMBL13533089 0.79 FAAH (0.42) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL745354 0.78 GSK3B (0.44) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL5441241 0.78 BRPF1 (0.40) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL26621513 0.78 MEN1 (0.44) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL3484140 0.78 DRD2 (0.40) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL746562 0.78 NOTUM (0.44) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL18069197 0.76 LMNA (0.45) BRPF1CCNB2CDK1CCNB1GSK3B
SCHEMBL751029 0.75 AADAT (0.47) KMT2AMEN1MAPTLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3464272-B1 NOVEL HETEROCYCLIC DERIVATIVES USEFUL AS SHP2 INHIBITORS JACOBIO PHARMACEUTICALS CO LTD (CN) 2021-12-08 EP disclosed