SCHEMBL2408111

SCHEMBL2408111

NC(=O)c1cccc(-c2cccc(N3CCC(CN(Cc4cscn4)C(=O)O)CC3)n2)c1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PRKD1 Q15139 1/20 0.37
PRKD2 Q9BZL6 1/20 0.37
SYK P43405 2/20 0.37
CNR1 P21554 2/20 0.37
PIM2 Q9P1W9 2/20 0.37
SMN1; SMN2 Q16637 2/20 0.36
MTOR P42345 2/20 0.36
CKS1B P61024 1/20 0.36
SKP1 P63208 1/20 0.36
SKP2 Q13309 1/20 0.36
PKM P14618 1/20 0.36
NPC1 O15118 1/20 0.36
RAB9A P51151 1/20 0.36
PIM1 P11309 2/20 0.35
FYN P06241 1/20 0.35
HTR1A P08908 1/20 0.35
HTR2A P28223 1/20 0.35
FFAR4 Q5NUL3 1/20 0.35
PDE10A Q9Y233 1/20 0.34
CCNT1 O60563 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2404007 0.92 CPT2 (0.35) PRKD1PRKD2SYKCKS1BSKP1
SCHEMBL2406016 0.92 SYK (0.38) PRKD1PRKD2SYKCNR1PIM2
SCHEMBL2407113 0.90 SMN1; SMN2 (0.44) CNR1PIM2SMN1; SMN2PIM1FYN
SCHEMBL2411489 0.88 CKS1B (0.42) CNR1CKS1BSKP1SKP2PKM
SCHEMBL2406060 0.87 DKK1 (0.42) CNR1PIM2SMN1; SMN2NPC1RAB9A
SCHEMBL2405635 0.87 PIM2 (0.36) CNR1PIM2CKS1BSKP1SKP2
SCHEMBL2406718 0.87 KMO (0.38) CNR1CKS1BSKP1SKP2FFAR4
SCHEMBL2407267 0.87 CKS1B (0.41) PRKD1SYKCNR1CKS1BSKP1
SCHEMBL2405902 0.86 FFAR4 (0.41) CNR1FFAR4
SCHEMBL2407614 0.86 FFAR4 (0.42) CNR1FFAR4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8912218-B2 Alkylthiazol carbamate derivatives, preparation thereof and therapeutic use thereof SANOFI (FR) 2014-12-16 US disclosed
US-20110212963-A1 ALKYLTHIAZOL CARBAMATE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF SANOFI-AVENTIS (FR) 2011-09-01 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110212963-A1 ALKYLTHIAZOL CARBAMATE DERIVATIVES, PREPARATION THEREOF AND THERAPEUTIC USE THEREOF MET, ALK, REL PRKD1 2512/4885PRKD2 3006/4885SYK 476/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.