SCHEMBL24089931

SCHEMBL24089931

O=S1(=O)Cc2cccnc2C1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 4/20 0.42
MEN1 O00255 3/20 0.42
SLC40A1 Q9NP59 5/20 0.35
CYP1A2 P05177 1/20 0.32
CYP2C19 P33261 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32
CA9 Q16790 1/20 0.32
S100A4 P26447 1/20 0.31
CDC25B P30305 1/20 0.31
TIPARP Q7Z3E1 1/20 0.31
TDP1 Q9NUW8 2/20 0.31
HTR3E A5X5Y0 1/20 0.31
HTR3B O95264 1/20 0.31
HTR3A P46098 1/20 0.31
HTR3D Q70Z44 1/20 0.31
HTR3C Q8WXA8 1/20 0.31
DRD2 P14416 1/20 0.31
DRD3 P35462 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL752924 0.82 DRD2 (0.35) KMT2AMEN1CYP1A2CYP2C19DRD2
SCHEMBL17902635 0.75 MEN1 (0.39) KMT2AMEN1SLC40A1CYP1A2CA12
SCHEMBL24089933 0.74 MEN1 (0.32) KMT2AMEN1
SCHEMBL29657671 0.71 KMT2A (0.64) KMT2AMEN1CYP1A2DRD2DRD3
SCHEMBL255964 0.71 KMT2A (0.64) KMT2AMEN1CYP1A2DRD2DRD3
SCHEMBL9252901 0.69 DPP8 (0.41) SLC40A1TIPARPDPP8DPP9FFAR4
SCHEMBL9256008 0.68 DPP8 (0.40) SLC40A1TIPARPDPP8DPP9
SCHEMBL7424121 0.67
SCHEMBL19152905 0.67 KMT2A (0.32) KMT2AMEN1HTR3EHTR3BHTR3A
SCHEMBL8348677 0.66

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20230312474-A1 PHENOL DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2023-10-05 US disclosed
US-20230312474-A1 PHENOL DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2023-10-05 US disclosed
EP-4206184-A1 PHENOL DERIVATIVE Sumitomo Pharma Co., Ltd. (JP) 2023-07-05 EP disclosed
US-11352366-B2 2-aminoquinazolinone derivative SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2022-06-07 US disclosed
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-16 US disclosed
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE SUMITOMO DAINIPPON PHARMA CO., LTD. (JP) 2021-12-09 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20210387967-A1 2-HETEROARYL AMINOQUINAZOLINONE DERIVATIVE CRKL, CLIC4, CLIC1 KMT2A 1451/4885MEN1 1679/4885SLC40A1 1436/4885
US-20230312474-A1 PHENOL DERIVATIVE TYR, NCOR1, BET1 KMT2A 356/4885MEN1 1330/4885SLC40A1 1178/4885
US-20210380598-A1 2-AMINOQUINAZOLINONE DERIVATIVE CNKSR1, HAX1, SLC26A3 KMT2A 967/4885MEN1 1282/4885SLC40A1 1929/4885
US-11352366-B2 2-aminoquinazolinone derivative CNKSR1, HAX1, SLC26A3 KMT2A 967/4885MEN1 1282/4885SLC40A1 1929/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.